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(1S,4S)-2-(2-chlorophenyl)-5-{2-[3-(trifluoromethyl)phenyl]acetyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
8-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-1H-1,3-benzodiazole-4-carboxamide
1-({3-[4-(2-hydroxyethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)azepan-2-one
3-[2-(dimethylamino)ethyl]-1-ethyl-8-(1H-indol-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1-[2-(3-fluorophenyl)ethyl]piperidin-2-one
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2,3-dimethoxy-N-(2-methoxyethyl)benzamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-3-cyclopropyl-N-methyl-1H-pyrazole-5-carboxamide
2-[3-(azepan-1-ylmethyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
5-chloro-2-hydroxy-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)benzamide
(4-{[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}oxan-4-yl)methanol
2-{4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
(4-methyl-5-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methanol
1-ethyl-4-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
(1S,5R)-3-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(4-benzylpiperidine-1-carbonyl)-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
7-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
2-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N,1-dimethyl-5-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrrole-2-carboxamide
2-{4-cycloheptyl-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-amino-4-(4-methyl-1H-imidazol-5-yl)-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
8-(6-aminopyridine-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-methylphenoxy)ethan-1-one
1-(5-fluoropyridine-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
methyl 2-[4-(6-methyl-2-oxo-1,2-dihydropyridine-3-amido)piperidin-1-yl]acetate
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-2-methylpyrimidin-4-amine
5-[4-(6-methyl-2-propylpyrimidin-4-yl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
1-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]cyclopropan-1-amine
2-[2-(3-chloro-4-methoxyphenyl)-4-methylphenoxy]acetamide
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide
2-(3-chlorophenoxy)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}thian-4-amine
8-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridin-3-amine
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
2-{[2-(methylsulfamoyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-fluorophenyl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-{5-cyclopropyl-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(thiophen-2-yl)pyrimidine
4-[2-(2-methoxyethyl)morpholin-4-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
5,6-dimethyl-3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
4-{[(4-fluorophenyl)methyl]amino}-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one