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(3aR,6aS)-1-oxo-2-propyl-5-(2-propylpyridine-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,2,3,4-tetrahydronaphthalene-2-carboxamide
(1S,5R)-3-(4-methylquinolin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-ethyl-1-methyl-3-{1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methoxypropan-1-one
(1R,5S,8S)-3-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-(3-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
5-{1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
N,N-diethyl-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
methyl (2S)-2-({2-[(2-methylphenyl)carbamoyl]ethyl}amino)-2-phenylacetate
8-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamido}phenyl)pentanamide
3-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N,N,15-trimethyl-13-oxo-9-phenyl-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-(cycloheptylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-1,3-thiazole-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-propoxypropanamide
1-[4-({3-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]-1H-1,2,4-triazole
2-(2-chloro-4-fluorophenoxymethyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
1-cyclohexyl-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
3-[(cycloheptylamino)methyl]-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-(2-methoxyethyl)-2-(pyridin-4-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1'-(5-methylpyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
3-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(1R,5R)-3-cyclobutanecarbonyl-6-{[4-(difluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
methyl 5-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,5R)-3-cyclobutanecarbonyl-6-(5-methylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-8-{[2-(furan-2-yl)phenyl]methyl}-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-[4-(1H-pyrazol-1-yl)butan-2-yl]thieno[2,3-d]pyrimidin-4-amine
1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
(3S,4R)-3-ethyl-4-methyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-ol
4-(1H-1,3-benzodiazol-1-yl)thiophene-2-carboxamide
N-(2-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)acetamide
diethyl({2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl})amine
4-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}morpholine
4-({4-[3-(4-fluoropiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
5-({3-[2-(dimethylcarbamoyl)ethyl]piperidin-1-yl}methyl)-2-hydroxybenzoic acid
N-{[3-(2-methoxyethoxy)phenyl]methyl}oxolane-3-carboxamide
4-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-(2-methoxyphenyl)-4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)piperazine
(3E)-1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pent-3-en-1-one
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})[2-(pyrrolidin-1-yl)ethyl]amine
N-benzyl-N-methyl-3-{[(pyridin-3-ylmethyl)amino]methyl}pyridin-2-amine
7-fluoro-3-({[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]amino}methyl)-1,2-dihydroquinolin-2-one