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4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
N-{[2-(1-methyl-1H-pyrazol-4-yl)phenyl]methyl}propanamide
1-ethyl-4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-{[4-methyl-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N'-(2-ethoxyphenyl)-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]propanediamide
3-[3-methyl-5-(1-methyl-4-phenylpiperidin-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(3R,4S)-4-cyclopropyl-1-(3,6-dimethylpyrazin-2-yl)pyrrolidin-3-amine
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-(trifluoromethyl)cyclopropane-1-carboxamide
3-[1-(5-chloropyridin-2-yl)piperidin-3-yl]-N,N-dimethylpropanamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-methoxy-6-({4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
5-[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-(2-methoxyethyl)-3-(propan-2-yl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,5-dimethyl-1-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
5-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-dimethyl-1H-pyrazole
5-({4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}methyl)-2-phenylpyrimidine
2-ethoxy-3-{[2-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}pyridine
2-(2H-1,3-benzodioxol-5-yl)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
8-[(2-ethylpyrimidin-5-yl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1,3-benzothiazol-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-fluorophenyl)-1,4-diazepane
4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}pyrimidine-5-carboxylic acid
1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
3-(4-hydroxyphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
4-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazole
3-methyl-8-{[3-(trifluoromethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-amino-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
8-[(3,4-dimethylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(2-chlorophenyl)-1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-cycloheptyl-3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
1-[(1-{[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]azepane
(1-methyl-1H-imidazol-2-yl)({1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl})methanol
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl 2-({3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}amino)benzoate
3-(4-chloro-1-methyl-1H-indole-2-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(3-oxo-3-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}propyl)piperidin-2-one
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)benzoic acid
pyridin-2-yl(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methanol
3-(4-acetylphenyl)-1-cyclohexyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
methyl 3-{4-[1-(dimethylamino)ethyl]phenyl}benzoate
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-4-yl)propan-1-one
N-[(2-methylphenyl)methyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrrol-1-yl)pentanamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-benzyl-N-methyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-3-amine