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2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-ethyl-N-methylacetamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(dicyclopropylmethyl)methylamine
3-(3,5-dimethylphenyl)-N-(2-methanesulfonylethyl)propanamide
(2E)-N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-(2-chlorophenyl)-N-(pyridin-2-ylmethyl)prop-2-enamide
3-[2-(3-methoxyphenyl)ethyl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(4-acetamidophenyl)methyl]-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
(5-{1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
2-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-3-methylpyridine
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
8-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(1R,7S)-3-(2-ethoxyethyl)-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1,3-thiazole
2-methoxy-2-phenyl-N-{1-[1-(prop-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
2-cyclopropyl-N-({1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)acetamide
(3R,4R)-4-amino-1-({3-ethoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)piperidin-3-ol
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(2-methoxyethyl)piperidine
5-tert-butyl-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1,3,4-oxadiazol-2-amine
ethyl 4-{1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-yl}piperazine-1-carboxylate
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(2-methylpiperidin-1-yl)-2-oxoacetamide
(3aS,6aR)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[2-methoxy-5-(methylcarbamoyl)phenyl]-4-(thiophen-2-ylmethyl)piperazine-1-carboxamide
2-(5-chloro-2-methoxyphenyl)-2-[methyl(1,2-oxazol-3-ylmethyl)amino]acetic acid
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2,3-dimethoxyphenyl)-2-(3-oxo-4-phenylpiperazin-1-yl)acetic acid
2-methoxy-N-(3-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}phenyl)benzamide
N-(3-hydroxypropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopentyl-N'-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]butanediamide
7-[(5-hydroxy-2-methoxyphenyl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-ethyl-N,N-dimethyl-6-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}pyrimidin-2-amine
N-methyl-N-[2-(2-methylphenyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
ethyl 1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
[2-(1,2,3,4-tetrahydroisoquinolin-5-yl)-1,3-thiazol-4-yl]methanol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-ethoxyethyl)piperidine-2-carboxamide
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
5-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrazine-2-carboxamide
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
5-fluoro-2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
3-[(3R,4S)-4-(dimethylamino)-1-[(2,3,4-trifluorophenyl)methyl]piperidin-3-yl]propan-1-ol
2-(2,3,4-trimethoxyphenyl)pyridine-4-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
1-cyclobutanecarbonyl-4-{5-[(4-methylpiperazin-1-yl)methyl]furan-2-carbonyl}-1,4-diazepane
1-[4-(2-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]aziridine-2-carboxylic acid
(3S,4R)-1-[(8-methylquinolin-5-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-{5-[3-(pyridin-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2-azaspiro[4.4]nonan-3-one
(4aS,7aR)-1-[3-(3-fluorophenyl)propanoyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione