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N-[(3-hydroxyphenyl)methyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
(2S,4S)-4-amino-1-[2-(2,4-dimethoxyphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
N-(5-propyl-1,3,4-thiadiazol-2-yl)-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]acetamide
6-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-N-methyl-3-({[2-(pyridin-4-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-(3-chloro-4-propanamidophenyl)-2-methoxypyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-(5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)-1,4-oxazepane
1-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}cyclohexan-1-ol
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-(pyridin-3-yl)propanamide
4-(hydroxymethyl)-1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperidin-4-ol
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-[2-(dimethylsulfamoyl)ethyl]urea
methyl 2-[N-methyl-1-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidin-4-yl)formamido]acetate
4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
3-cyclopropyl-1-[2-(piperidin-1-ylmethyl)phenyl]-3-(thiophen-3-ylmethyl)urea
N-[1-(carbamoylmethyl)piperidin-4-yl]-4-(4-chlorophenyl)butanamide
N-benzyl-2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
3-(1-{1-[(2S)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-chlorophenyl)urea
2-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}azetidin-3-yl)pyridine
(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]isoquinoline
4-amino-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-(3-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-ethyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(pyridin-4-ylmethyl)benzamide
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
(2S)-3-(1H-indol-3-yl)-2-{[1-(pyrimidin-2-yl)piperidin-4-yl]amino}propan-1-ol
N-[(3-methoxyphenyl)methyl]-3-[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]propanamide
3-methyl-3-{[3-(methylsulfanyl)phenyl]methyl}-1-[4-(morpholin-4-ylmethyl)phenyl]urea
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
4-benzyl-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
4-(3-hydroxy-3-methylbutyl)-N-(oxan-3-yl)benzamide
9-[(3-chlorophenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-fluorophenyl)-6-[2-(1H-indazol-1-yl)acetyl]-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 1-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}pyridine
4-(4-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
9-(8-chloroquinolin-2-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
(3R,4S)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3,4-dimethylpiperidin-4-ol
N-(propan-2-yl)-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-8-{[3-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
({5-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
1-(3-methoxypropyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methylpiperidin-3-amine
(3S,4S)-4-cyclopropyl-1-(3-sulfamoylbenzoyl)pyrrolidine-3-carboxylic acid
N-(3-chloro-4-methoxyphenyl)-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}propanamide
1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
1-(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one