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[(4-methanesulfonylphenyl)methyl](methyl)(quinolin-5-ylmethyl)amine
2-(piperidin-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
2-(5-acetylthiophen-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
(3R,4S)-4-cyclopropyl-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
(2R)-2-[(2-benzyl-1,3-thiazol-4-yl)formamido]-3-(pyridin-4-yl)propanoic acid
1-(furan-2-ylmethyl)-4-[(3-methylphenyl)methyl]-1,4-diazepane-6-carboxylic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-5-phenyl-1H-pyrrole-2-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
(2S)-6-amino-2-[2-(2,3,6-trimethylphenoxy)acetamido]hexanoic acid
4-(1-phenyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propan-2-yl]pyrimidin-2-amine
1-{2-[3-phenyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
1-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)urea
4-{4-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
N-methyl-2-(phenylformamido)-N-(quinolin-5-ylmethyl)acetamide
1-(7-fluoro-4-methylquinolin-2-yl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N,N-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]aniline
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]benzonitrile
2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-({1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
2-[ethyl(methyl)amino]-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N4-ethyl-N2-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
4-hydroxy-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazine-1-sulfonamide
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-2-(phenylamino)pyrimidine-5-carboxamide
2-methyl-3-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
2-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-(2-fluorophenyl)-1H-pyrrole
(1r,4r)-4-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}cyclohexan-1-ol
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-benzyl-2-(4-methoxyphenyl)piperidine-1-sulfonamide
1-(3-chlorophenyl)-4-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(4,4,4-trifluorobutan-2-yl)piperidin-4-yl]oxy}benzamide
(4aR,8aR)-4-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-octahydro-2H-1,4-benzoxazine
N-cyclopropyl-3-(2-methylpropyl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
2-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}thiophen-3-amine
methyl (2S,4R)-1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-4-hydroxypyrrolidine-2-carboxylate
5-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
3-methyl-5-{4H-thieno[3,2-b]pyrrol-5-yl}-1H-1,2,4-triazole
ethyl 4-[3-(1H-imidazol-2-yl)benzamido]piperidine-1-carboxylate
2-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyridine-3-carboxamide
2-(2-ethylpyrimidin-5-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)quinoline-4-carboxamide
3-({[1-(5-propylthiophene-3-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-methyl-N4-{[1-(2-phenylethyl)piperidin-4-yl]methyl}pyrimidine-4,6-diamine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
4-[(3-carbamoyl-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-2,6-dimethylphenyl acetate