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2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[4-(oxolan-2-yl)butyl]acetamide
N2-(2-methoxyethyl)-N4-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-2-(3-phenylpropyl)morpholine
2-{1-[(2-fluorophenyl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
7-(1H-1,2,3-benzotriazole-5-carbonyl)-2-oxa-7-azaspiro[4.5]decane
N-(3-chloro-2-methylphenyl)-3-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropanamide
7-[(3-methoxyphenyl)methyl]-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-({2-[(benzenesulfonyl)methyl]phenyl}methyl)azepan-3-amine
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
9-(3-chloro-5-methoxybenzoyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
5-[1-(3-methylbut-2-en-1-yl)pyrrolidin-2-yl]-N-[2-(methylsulfamoyl)ethyl]thiophene-2-carboxamide
4-(4-chlorophenyl)-N-(oxan-4-yl)butanamide
(3S,4R)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-methoxypyrimidine
4-(2H-1,3-benzodioxol-5-yl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2H-1,3-benzodioxole-5-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1,3-dimethyl-5-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
2-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]-4-hydroxyquinoline-6-carboxamide
1-(5-chloro-2-methoxybenzoyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
methyl[1-(1,2-oxazol-3-yl)ethyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-(furan-3-yl)-1-[(1R)-1-(4-methoxyphenyl)ethyl]-1H-imidazole
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-[(oxolan-3-yl)sulfamoyl]-N-(pyrimidin-4-ylmethyl)benzamide
1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-(pyrrolidine-1-carbonyl)pyridine
2-(1-methyl-1H-imidazol-2-yl)-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]benzamide
(4aR,7aS)-1-acetyl-4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 5-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(5-fluoropentyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
9-(cyclopropylmethyl)-4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-methoxyphenyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-({3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)quinoline
2-(4-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}phenoxy)pyrimidine
(4aS,8aR)-1-butyl-6-(4-methoxycyclohexanecarbonyl)-decahydro-1,6-naphthyridin-2-one
3-[(1-acetylpiperidin-4-yl)amino]-N-(2,3-dihydro-1H-inden-2-yl)-5-[(propan-2-yl)sulfamoyl]benzamide
1-[(3-fluorophenyl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylimidazo[1,2-a]pyrimidine
7-(4-chlorophenyl)-2-(pyridin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-1-(4-methylphenyl)piperazin-2-one
1-cyclohexyl-3-hydroxy-4-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(pyrazin-2-yl)propan-2-yl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
2-(4-methylpentyl)-4-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]morpholine