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N-{1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}methanesulfonamide
{4-[(3-chloro-1H-indol-2-yl)methyl]-1-methylpiperazin-2-yl}methanol
4-methyl-9-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetyl}-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
1-(2,3-dihydro-1H-inden-4-yl)-3-(oxan-4-yl)-5-[(2R)-pyrrolidin-2-yl]-1H-1,2,4-triazole
4-{[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
N-[4-fluoro-3-({[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]carbamoyl}amino)phenyl]acetamide
2-({6-[2-(pyridin-2-yl)-1H-imidazol-1-yl]quinazolin-4-yl}amino)ethan-1-ol
3-{5-[(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
{3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-oxopropyl}urea
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(phenylsulfanyl)acetamide
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N-(3-cyclopentylpropyl)-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-phenyl-1,2,4-oxadiazole
ethyl 4-(1-benzofuran-3-carbonyl)piperazine-1-carboxylate
N-butyl-1-cyclohexyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
2-(4-{[4-(5-methylfuran-2-yl)phenyl]methyl}morpholin-3-yl)acetic acid
3-[3-(3-methoxypropyl)piperidine-1-carbonyl]benzene-1,2-diol
(3aS,6aS)-1-methyl-5-[(5-propylfuran-2-yl)methyl]-octahydropyrrolo[3,4-b]pyrrole
2-(2-ethyl-1H-imidazol-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
N-[(3R,4R)-1-[2-(4-chlorophenyl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
1-{1-[(4-ethynylphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
14-(4-hydroxyquinolin-2-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(2-fluoro-5-methylphenyl)-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
5-fluoro-2-{1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-methoxy-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}acetamide
methyl 2-[benzyl(methyl)sulfamoyl]-6-(2-ethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
[(1R,3S,3aS,6aR)-1-(1H-indol-3-ylmethyl)-5-methyl-3-(5-methylfuran-2-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2,5-dichloro-N-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-hydroxy-N-methyl-1,2-oxazole-5-carboxamide
(2R,6S)-2,6-dimethyl-4-(5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)morpholine
[(3R,5R)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
4-(2-fluorophenoxy)-1-(oxane-2-carbonyl)piperidine-4-carboxylic acid
N-methyl-2-(2-methylphenyl)-N-[1-(pyridin-4-yl)ethyl]benzamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(3-methoxyphenyl)azetidine
N'-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-N-methylbutanediamide
5-[(dimethylamino)methyl]-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}furan-2-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
5-fluoro-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyrimidin-4-amine
N-{1-[1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidin-4-ol
N-[(1S)-1-(3-benzyl-1H-1,2,4-triazol-5-yl)-3-(methylsulfanyl)propyl]acetamide
(1S,5R)-3-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4,6-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
[(2-methoxyphenyl)methyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})propylamine
[5-(1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
4-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)pyridine-3-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,N-dimethyl-6-(trifluoromethyl)pyrimidin-2-amine