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ethyl 4-[(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-(5-methanesulfonamido-2-methylphenyl)urea
5-(azepane-1-carbonyl)-N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-ethyl-1H-pyrazole
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[3-(2-methoxyphenyl)propyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-{3-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
(1R,5S)-8-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-3,8-diazabicyclo[3.2.1]octane
1-acetyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}piperidine-4-carboxamide
1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethan-1-amine
(2S,4R)-4-amino-N-methyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]pyrrolidine-2-carboxamide
2-[4-(5-acetylpyridin-2-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
4-{[4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl]methyl}phenol
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[3-(pyrrolidin-1-ylmethyl)phenyl]methyl})amine
(3aR,6aR)-2-(dimethylcarbamoyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
2-{3-[(4-acetylpiperazin-1-yl)methyl]phenyl}-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
5-{2-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}-2-methoxy-N-methylbenzamide
N-cyclopropyl-5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
3-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-amine
3-(4,4-difluoropiperidine-1-carbonyl)-4-fluorobenzene-1-sulfonamide
N,3,5-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
2-(3,4-dichlorophenyl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholine
4-ethyl-3-(1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(pyridin-3-yloxy)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
2-(methylamino)-N-[(1-methylpiperidin-3-yl)methyl]benzamide
5-(2-chloro-4-fluorophenyl)pyridin-2-amine
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(3-fluorobenzoyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-6-methyl-3-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(azepan-1-yl)-2-phenylethyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1,4-dimethyl-2-{[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazine
7-methyl-2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-2,7-diazaspiro[4.5]decan-6-one
2-(5-fluoro-2-methylphenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
2-(6-aminopyridin-3-yl)-2-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}acetic acid
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(3-methylphenoxy)azetidin-1-yl]pyrimidine
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methyloxetan-3-yl)methyl]acetamide
4-{1-[6-(1H-pyrazol-3-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
3-(2,4-dimethoxybenzoyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
4-(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)phenol
7-(cyclopropylmethyl)-2-(propane-2-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2,2-difluoroethyl)-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-chloro-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-propanamidobenzamide
4-[methyl(1,2-oxazol-5-ylmethyl)sulfamoyl]-N-[(3S)-pyrrolidin-3-yl]benzamide