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N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-oxopyrrolidin-2-yl)acetamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(piperidin-4-yl)propanamide
2-(adamantan-1-yl)-4-hydroxy-N-(5-hydroxypentyl)pyrimidine-5-carboxamide
1-cyclopentyl-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
5-{1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-3-hydroxypropanamide
7-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
9-(4,6-dimethylpyridine-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidin-2-amine
1-(2-chlorophenyl)-4-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperazin-2-one
7-(4-chlorophenyl)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
butyl({[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl})methylamine
1-(2,5-dichlorophenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
N-[2-methoxy-5-({[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}amino)phenyl]acetamide
4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-1-(2-methylpropyl)piperidine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(dimethylamino)-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-(3-methylphenyl)acetamide
2-(cyclopropylmethyl)-9-[2-(dimethylamino)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
2-({[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}methoxy)acetamide
(3S,5R)-1-benzyl-N3-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
3,6,7-trimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-({[3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
(2S,4S)-4-amino-N,N-diethyl-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)pyrrolidine-2-carboxamide
2-(4-hydroxybutyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidin-2-one
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
1-(3-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenyl)ethan-1-one
1-cyclobutanecarbonyl-4-(1H-imidazol-2-ylmethyl)-1,4-diazepane
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]thiophen-3-amine
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
3-(4-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
4-(3-fluorophenyl)-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
(3aR,6aR)-2-(2,5-dimethylfuran-3-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
4-[4-methyl-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
2-{1-[(3,4-difluorophenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
4-(4-fluorophenoxy)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
2-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-5-methoxypyridin-4-ol
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(oxane-4-carbonyl)piperidine
{3-[(2-fluorophenyl)methyl]-1-[4-(trifluoromethyl)benzoyl]piperidin-3-yl}methanol
8-[2-(2,4-dimethoxyphenyl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{[methyl({[3-(2-{4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
N-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)benzamide