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5,6-dimethyl-N4-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidine-2,4-diamine
5-(methoxymethyl)-N-(4-{5-methyl-4-[(2-phenoxypropanamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-2-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-(2-methoxyethyl)-2-(methylamino)-N-[(4-methylphenyl)methyl]pyridine-3-carboxamide
1-{1'-[2-(3-hydroxyphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3R,4S)-3-[2-(3-fluorophenoxy)acetamido]-4-propylpyrrolidin-1-yl]propanoic acid
2-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
2-tert-butyl-8-(2,7-dimethylquinoline-4-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(2,4-difluorophenyl)-1-[2-(dimethylamino)ethyl]-6-(oxan-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{[(1R,5S,6S)-3-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
(2R,3R)-3-[4-(2-fluorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(1H-pyrazol-1-yl)butanamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetamide
N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
(3S,4S)-4-cyclopropyl-1-{[(2-methylphenyl)methyl]carbamoyl}pyrrolidine-3-carboxylic acid
(2R,3R,6R)-5-(2,4-dimethylpyrimidine-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-[(pyrimidin-4-ylmethyl)amino]pyridine-3-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
5-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-4,6-dimethyl-2H-pyran-2-one
3-[(3R,4S)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-[3-({[2-methoxy-2-(thiophen-2-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
2-[1-(3-methylbutyl)-2,4-dioxo-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-({7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
[(3R,5S)-1-[(5-ethylpyridin-2-yl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-[2-(2-chloro-6-methoxyphenyl)-4-methylphenyl]propanamide
2-[(2-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
(3S,4S)-4-[4-(pyrazin-2-yl)piperazin-1-yl]-1-(thiophen-3-ylmethyl)pyrrolidin-3-ol
N-(cyclopropylmethyl)-3-[(2-methanesulfonylethyl)sulfamoyl]benzamide
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
N-(3-chlorophenyl)-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butanamide
1-{4-[3-(1H-pyrazol-3-yl)phenyl]thiophen-2-yl}ethan-1-one
N-cyclopropyl-1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(2-methylphenyl)-2-{4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}acetamide
3-{2-[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}piperidin-3-yl)morpholine
7-(cyclopropylmethyl)-2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
6-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
N-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)acetamide
2-[1-(pyrazin-2-yl)propan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[3-(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}pyridine
methyl 3-benzamido-5-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
(3ar,6ar)-N-(2-propoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)-4-methylphenol
3-[(2-fluorophenyl)methyl]-5-(oxan-4-yl)-1,2,4-oxadiazole