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2-[4-(pyridin-2-yl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
N-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
(7S,8aS)-7-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-(cyclopropylmethyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-6-(2-methoxyphenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyridine-3-carboxamide
7-(3,5-dimethoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
4-{1-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl](2-phenylpropyl)amine
1-cyclopropanecarbonyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(4S)-3,3,4-trimethyl-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-ol
2-{1-[(8-methoxy-2H-chromen-3-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
3-[1-({1-[(thiophen-2-yl)carbamoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]propanoic acid
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
9-(2-hydroxy-3-methoxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carbonyl}-1λ6-thiomorpholine-1,1-dione
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
(2R)-2-{[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}-4-methylpentanamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(1-propylpiperidin-4-yl)piperidine
N-benzyl-5-(2,5-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-{[4-methoxy-3-(thiophen-3-ylmethoxy)phenyl]methyl}-5,7-dimethyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-{5-[(3-fluoro-2,4-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
6-(4-fluorophenyl)-7-methyl-N-(2-methylbutyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-4-(piperidin-1-ylmethyl)benzamide
methyl 3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N,N-dimethyl-5-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}pyrimidin-2-amine
(3S,4S)-4-cyclopropyl-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(5-ethyl-1,2,4-oxadiazol-3-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(3-fluorophenyl)benzoyl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyrimidin-4-amine
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
1-[4-chloro-3-(trifluoromethyl)phenyl]-4-(oxane-4-carbonyl)piperazine
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
N-(1-methoxybutan-2-yl)-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
8-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
(1-{[1-(2,3-difluoro-4-methoxybenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methylphenol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-3-yl)propanamide
2-{4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazin-1-yl}pyrazine
methyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})[(4-phenoxyphenyl)methyl]amine
N,N-dimethyl-5-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)pyridin-2-amine
5-({2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}methyl)-N,N-dimethylpyridin-2-amine
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-4-yl)pyridine
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-1-(2-methoxyethyl)-3-(prop-2-en-1-yl)urea
N-cyclopropyl-4-methoxy-2-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-cyclopentyl-N-[(2,3-dimethoxyphenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
7-(cyclopropylmethyl)-2-(4-phenoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one