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N-ethyl-N-(1-hydroxypropan-2-yl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
3-methyl-5-(3-phenylpropyl)-1H-1,2,4-triazole
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
(2S,4R)-4-amino-N-methyl-1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}pyrrolidine-2-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-(6-chloro-2-methylquinoline-4-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]benzonitrile
N-({8-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
N-[(2-ethoxyphenyl)methyl]-N-{[5-(oxan-2-yl)furan-2-yl]methyl}cyclopropanamine
(4aS,7aR)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-4-yl)pyridin-2-amine
1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(thiophen-3-yl)propan-1-one
N-[(3R,4R)-3-hydroxy-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl]pyridine-2-carboxamide
ethyl 4-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}piperazine-1-carboxylate
1-(2-fluorophenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}cyclopropane-1-carboxamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(methanesulfonylmethyl)piperidine
4-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-3-(1H-pyrrol-1-yl)benzamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]benzamide
5-amino-4-chloro-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazole-3-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
methyl 3-(2-methylbutanamido)-5-{[1-(methylsulfanyl)propan-2-yl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[3-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-6-methylpyridine-2-carboxamide
4-hydroxy-N-[1-(pyrazin-2-yl)propan-2-yl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-(azetidine-1-sulfonyl)-N-methyl-N-(thian-4-yl)benzamide
5-ethyl-2-methyl-4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
2-ethyl-N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}butanamide
5-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridine-2-carbonitrile
1-{2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-methyl-1,2-dihydroquinolin-2-one
4-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperazine-1-carboxamide
1-(2-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
4-(2H-1,3-benzodioxol-5-yl)-3-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(3-acetamidophenyl)-2H-1,3-benzodioxole-5-carboxamide
5-ethyl-1'-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[5-(2,3-dihydro-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
(3R,4S)-3,4-dimethyl-1-[(2-phenylphenyl)methyl]piperidin-4-ol
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[(2E)-3-(4-methoxyphenyl)prop-2-enamido]ethyl}-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-ethyl-4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
1-[3-(azepane-1-carbonyl)-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]-4-(4-chlorophenyl)piperidin-4-ol
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-(dimethyl-1,3-thiazol-5-yl)acetamide
N-[(2R,4R,6S)-2-cyclohexyl-6-[1-(propan-2-yl)piperidin-4-yl]oxan-4-yl]acetamide
1-(furan-2-carbonyl)-4-[6-(methoxymethyl)pyridine-2-carbonyl]-1,4-diazepane
[4-(6-cyclopropylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
2-[1-(2-methoxybenzenesulfonyl)pyrrolidin-3-yl]benzoic acid
{3-[(4-fluorophenyl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl}methanol
3,5-dimethoxy-2-({methyl[(1-methylpiperidin-3-yl)methyl]amino}methyl)benzoic acid