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2-cyclopropyl-N-ethyl-N-[2-(morpholin-4-yl)ethyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-(2-fluorophenyl)-5-(2-methoxy-5-methylbenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
4-[3-(2-methoxyphenoxy)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
6-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carboxylic acid
4-methyl-6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
4-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one
5-(morpholin-4-yl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]-2,3-dihydropyridazin-3-one
6-(2-chlorophenyl)-N-(2-fluoroethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2-aminoethyl)-N-benzyl-N-[2-(dimethylamino)ethyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[2-(furan-2-yl)ethyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(4-phenyl-1H-pyrazol-1-yl)acetamide
3-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
4-(4-methoxy-2-methylphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
5-{2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
(4aS,7aR)-1-(5-methylpyridine-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
3-ethyl-2-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1H-indole
5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyrimidine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-4-(propan-2-yl)piperazine
(1S,6R)-9-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
dimethyl({2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl})amine
2-chloro-N-ethyl-4-fluoro-N-[2-(morpholin-4-yl)ethyl]benzamide
2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
N-(3-methoxyphenyl)-3-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]propanamide
3-(1H-indazol-7-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
4-fluoro-3-[3-methyl-5-(4-propylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
ethyl 3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carboxylate
6-(2,5-dimethylbenzoyl)-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(5-propyl-1,3,4-oxadiazol-2-yl)amino]methyl}pyrrolidin-2-yl]methanol
N-(3-chlorophenyl)-3-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)propanamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
3-(2-methoxyphenyl)-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}propan-1-one
5-[1-(1-benzofuran-2-ylmethyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(pyridin-3-ylmethyl)amino]pyridine-3-carboxamide
N-ethyl-1-(2-methoxyacetyl)-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-[(5-methylhex-5-en-2-yl)amino]-N-(2-methylphenyl)acetamide
8-(1H-imidazol-4-ylmethyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 3-(2-phenoxyethyl)piperidine-3-carboxylate
dimethyl({2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-1-(3-methylthiophen-2-yl)ethyl})amine
N-[2-(oxolan-3-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{[3-(dimethylamino)propyl](methyl)amino}-2-(4-methoxy-3,5-dimethylphenyl)acetic acid