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[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
N-(adamantan-2-yl)-6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-methyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)furan-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-(3-methylpyridin-4-yl)piperazin-1-yl]methyl}piperidin-2-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(4-methylphenyl)methyl]benzamide
6-cyclopropyl-2-[4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
1-methyl-9-(6-phenoxypyridin-3-yl)-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
1-{2-[3-(2-methoxyethyl)-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
(1R,4S)-2-[2-(5-chloro-2-methoxyphenyl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
2-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]acetic acid
3-({1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(cyclobutylmethyl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)propanamide
7-[2-(2-methylphenyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-3-[({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amino)methyl]benzamide
N-[5-(4-phenyl-1H-imidazol-5-yl)pyrimidin-2-yl]benzenesulfonamide
2-[4-(4-methanesulfonylphenyl)-6-methylpyrimidin-2-yl]phenol
(5S,9aS,9bS)-5-(4-methoxy-2,3-dimethylphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-tert-butyl-5-oxopyrrolidine-3-carboxamide
N-(3-hydroxypropyl)-2-(2-oxopyrrolidin-1-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(propan-2-ylsulfanyl)ethyl]acetamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole-5-carboxamide
2-amino-6-[4-fluoro-2-(trifluoromethyl)phenyl]-4-(oxolan-3-yl)pyridine-3-carbonitrile
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
(3aR,7aS)-2-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-cyclohexyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)pent-4-enamide
2-(2,3-dimethylphenyl)-N,N-dimethylpyridine-3-carboxamide
9-methoxy-4-[(1-methyl-1H-imidazol-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[1-cyclopentyl-4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-2-yl]ethan-1-ol
1-phenyl-2-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)ethane-1,2-dione
5-{[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2,2-dimethylbutan-1-one
1-(2,3-dihydro-1H-indene-1-carbonyl)-3-(2-methoxyphenoxy)azetidine
N-methyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
N-methyl-2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholin-3-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
N-[1-(2,3-dihydroxypropyl)piperidin-4-yl]methanesulfonamide
1-[(2-fluorophenyl)methyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6-oxopiperidine-3-carboxamide
5-(2-chloro-4-fluorophenyl)pyridine-3-carboxamide
6-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
3-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepane-1-carbonyl]benzonitrile
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
5-cyano-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
1-(cyclopropylmethyl)-4-(3,5-difluoropyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
methyl N-{[(2S,4S)-1-(1-benzoxepine-4-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}carbamate
1-{2-hydroxy-3-[2-methoxy-4-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
(3S,5S)-1-benzyl-N-[(3-chlorophenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine