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1-ethyl-5-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-[5-(5-chloro-2-methoxypyridin-4-yl)furan-2-carbonyl]morpholine
2-{1-[(2-methylphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
{4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenyl}methanol
(1S,9R)-11-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3,3-dimethyl-1-[(3S,4R)-1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-[1-(cyclopropylmethyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(2-hydroxyethyl)-9-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-5-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2,5-dimethyl-N-[(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-3-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylcyclohexanecarboxamide
(1R,5S,6S)-6-[1-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-3-azabicyclo[3.1.0]hexane
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-methyl-2-(3-{1-[3-(pyridin-3-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyridine
2-methyl-1-[4-({2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]propan-1-one
6-[2-(dimethylamino)phenyl]-N-methylpyridine-2-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
1-(4-chlorophenyl)-3-(2,2-dimethyloxan-4-yl)-3-ethylurea
4-[(dimethylamino)methyl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]azepan-4-ol
1-(naphthalen-1-yl)-3-[3-(oxolan-3-yl)propyl]urea
3-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]quinoline
4-[(4,5-dimethylfuran-2-yl)methyl]-2-[(4-methoxyphenyl)methyl]morpholine
4,4,4-trifluoro-3-[(3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid
N-[(5-methoxy-1H-indol-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1-(pyridin-2-yl)piperidine-3-carboxamide
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
(3S,4S)-1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-methylpiperidine-3,4-diol
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amine
2-(2-butyl-1H-imidazol-4-yl)-1-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-imidazole
N-benzyl-1-(2-hydroxyethyl)-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
8-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
8-fluoro-N-[2-(1H-imidazol-4-yl)ethyl]quinoline-2-carboxamide
4-({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}amino)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
1-(1-benzylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethylpyridine-4-carboxamide
1-{6-hydroxy-4-[2-(phenylsulfanyl)ethyl]-1,4-diazepan-1-yl}ethan-1-one
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-propoxyethan-1-one
1-[(4-chloro-3-fluorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(1H-imidazol-4-ylmethyl)-4-(oxane-4-carbonyl)-1,4-diazepane-6-carboxylic acid
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}butanamide
5-[1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-2-yl]-N-(1-methyl-1H-1,2,4-triazol-3-yl)thiophene-2-carboxamide
6,7-dimethoxy-2-(4-methylthiophen-3-yl)quinazolin-4-amine
2-[3-(pyrrolidin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-methoxyacetyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
5-[2-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-2-oxoethyl]-3-propylimidazolidine-2,4-dione
1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol