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1-methyl-3-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indole
4-(1H-pyrazol-4-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]butan-1-one
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
3-(1-ethyl-1H-pyrazol-4-yl)-1-{2-[methyl(phenyl)amino]ethyl}urea
1-{1-[(4-ethynylphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2,5-dimethyl-N-[(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-3-carboxamide
1-[(3S,4S)-3-hydroxy-4-(thiomorpholin-4-yl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
5,8-difluoro-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydroisoquinoline
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(3-methylthiophen-2-yl)ethyl]furan-2-carboxamide
1-{3-[(2,2-dimethylmorpholin-4-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
ethyl 4-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}piperidine-1-carboxylate
3-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-[(3R,4S)-4-(propan-2-yl)-1-(pyrazin-2-yl)pyrrolidin-3-yl]piperidine-1-sulfonamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
4-(4-methoxyphenyl)-2-methyl-3-oxo-N-pentylpiperazine-1-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(thiophen-2-ylmethyl)amine
2-acetyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-2-methylpyridine
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
N-[(2S,4R,6R)-2-(4-tert-butylphenyl)-6-(propan-2-yl)oxan-4-yl]acetamide
1-(furan-3-carbonyl)-4-(quinolin-2-yl)-1,4-diazepan-6-ol
N-(2-{7-[(4-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)acetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinoline-5-carboxamide
8-cyclopropanecarbonyl-2-[(3-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-2-carboxamide
2-[4-benzyl-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl]-N-cyclopropylacetamide
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
1-(4-{[4-(methylamino)butyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(3-oxopiperazin-1-yl)pyridine-3-carboxamide
4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(2R,3R,6R)-5-(2-ethylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-N-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-chloro-2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-phenylpropyl)-1H-1,2,3-triazole
7-chloro-4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
dimethyl({[5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)thiophen-3-yl]methyl})amine
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-{2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
2-methyl-6-({4-[4-(piperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
2,2-dimethyl-6-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-one
4-{[(3-ethoxyphenyl)methyl]amino}-1-[(4-fluorophenyl)methyl]pyrrolidin-2-one
4-(4-chloro-2-fluorobenzoyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
N-ethyl-N,8-dimethyl-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide