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3-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)pyridine
1-(cyclohexylmethyl)-4-[(4-ethyl-5-methylpyrimidin-2-yl)amino]pyrrolidin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-fluoro-2-methoxybenzoyl)pyrrolidin-3-yl]methanol
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4-methyl-2-(propan-2-yl)pyrimidine
(3aR,6aS)-2-methyl-5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
(3aS,6aS)-2-cyclopropanecarbonyl-5-(5-methoxyfuran-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-(thiophen-2-yl)butanamide
[5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
1-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-4-(pyridin-4-yl)piperazine
ethyl 1-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}-4-cyclopentylpiperazine
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-(oxolan-2-ylmethyl)-7-(propan-2-yl)-N-(thiophen-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenyl)acetamide
2-(4-methoxy-2-methylphenyl)-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
[(3R,4R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-(1-ethyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
methyl N-{2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}carbamate
2-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)-4-(methylsulfanyl)butanoic acid
2-(5-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}furan-2-yl)benzonitrile
8-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,3-dihydro-1H-indene-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]oxane-4-carboxamide
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-3-(methylsulfanyl)propanamide
4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine-1-carbaldehyde
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-(dimethylamino)-7-(2-hydroxy-4-methylbenzoyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(4-methoxybutyl)-4-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperazine
N-(1,4-dioxan-2-ylmethyl)-4-fluoro-3-methoxybenzamide
3-hydroxy-1-(2-methoxyethyl)-3-{[(thiophen-3-ylmethyl)amino]methyl}piperidin-2-one
3-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
4-[(3,4-difluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-methyl-1,4-diazepan-5-one
1-(6-tert-butyl-2-oxo-2,3-dihydropyrimidine-4-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(3S,4R)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-ethyl-4-methylpiperidin-4-ol
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-1,2,3-thiadiazole-4-carboxamide
7-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(methylamino)ethyl]-1,3-oxazole-4-carboxamide
2-methyl-5-phenyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-methyl-2-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1H-1,3-benzodiazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-hydroxyethyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
6-[({[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
4-(hydroxymethyl)-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}azepan-4-ol
3-(3-{4-[2-(trifluoromethyl)phenyl]-1H-1,2,3-triazol-1-yl}propyl)pyridine