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(3S,5R)-1-(1H-imidazol-2-ylmethyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
5-(2-methylpropyl)-1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S)-1-benzyl-N-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-amine
5-(methoxymethyl)-N-(3-methyl-1-{7-propyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
(3E)-2-[4-(2-methoxyethoxy)piperidin-1-yl]-4-phenylbut-3-enoic acid
5-{[(2,3-dimethoxyphenyl)methyl]amino}-1-ethyl-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{2-[2-methoxy-6-(1-methyl-1H-1,3-benzodiazol-2-yl)phenoxy]ethyl}dimethylamine
2-(furan-2-yl)-N-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyrrolidine-1-carboxamide
1-{2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carbonyl}piperidine-3-carboxamide
5-(2-methoxyphenoxymethyl)-N-propyl-1H-pyrazole-3-carboxamide
2-methoxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-methylpropan-1-one
3-cyano-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]benzamide
N-ethyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrimidin-2-amine
3-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-N-(2,5-dimethoxyphenyl)propanamide
1-(oxolan-2-ylmethyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5,6,7,8-tetrahydroquinazolin-2-amine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
3,5-dichloro-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N,4-dimethylbenzamide
(2S,4R)-4-(3-cyanobenzamido)-N-[(1-hydroxycyclohexyl)methyl]pyrrolidine-2-carboxamide
3,5-dimethyl-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-indole-2-carboxamide
5-(2-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[phenyl(pyridin-4-yl)methyl]piperidine-4-carboxamide
N-(1,3,4-thiadiazol-2-yl)-3-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}benzamide
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N-(propan-2-yl)pyridine-4-carboxamide
(2S,4R)-4-[4-({[(4-fluorophenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
1-(2-chlorophenyl)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethan-1-ol
3-(4-methoxyphenoxymethyl)-1-(5-methyl-1,2-oxazole-4-carbonyl)piperidine
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(3-hydroxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(4-hydroxyphenyl)-N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-(2-chloro-4-fluorobenzoyl)piperidine
N-ethyl-2-{4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazin-1-yl}acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]urea
2-(3-methyl-4-{[3-(3-methylphenyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(3,5-difluorophenyl)methyl]-1H-pyrazole-4-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-2-(furan-2-yl)-2-oxoacetamide
1-{1-[3-(ethylsulfanyl)propanoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-(2-chlorophenyl)-N-[(2S)-2-hydroxypropyl]-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-propyl-4-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]sulfamoyl}benzamide
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-phenyl-7-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N,4-dimethyl-2-(piperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidine-5-carboxamide
(3S,4R)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
4-{1-[2-(2,4-dimethoxyphenyl)-1H-imidazol-1-yl]propyl}pyridine
3-(4-benzyl-1H-pyrazol-5-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine