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methyl 6-{[2-(4-fluorophenyl)-3-oxopiperazin-1-yl]methyl}pyridine-2-carboxylate
4-[(2,4-dimethoxyphenyl)methyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]propanamide
methyl 6-(4-{2-[(1-benzylpyrrolidin-3-yl)carbamoyl]ethyl}piperidin-1-yl)pyridine-3-carboxylate
3,5-difluoro-2-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]pyridine
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N,N-dimethyl-4-oxobutanamide
N,5-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
3-{[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzoic acid
ethyl 4-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxylate
(3aS,6aR)-5-(1-benzofuran-2-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{2-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3-benzotriazole
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]naphthalene-1-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyrimidin-4-ylmethyl)acetamide
(2S,4R)-4-hydroxy-N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)pyrrolidine-2-carboxamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(1-methyl-1H-pyrrol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)morpholine-2-carboxamide
9-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(benzylsulfamoyl)({1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl})amine
(2S,4R)-N-methyl-1-(naphthalen-1-ylmethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
N-methyl-4-{[(3-methylthiophen-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}benzamide
N-(4-chloro-2-methoxy-5-methylphenyl)-2-[(methylcarbamoyl)methyl]-3-oxopiperazine-1-carboxamide
2-benzyl-8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-6-(3-propyl-1H-pyrazole-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
(1S,5R)-3-benzoyl-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
9-{[4-(2-aminoethyl)phenyl]methyl}-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[3-(5-chlorothiophen-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
(2S,4R)-4-amino-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(2-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenoxy)ethan-1-ol
3-({2-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-{4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methyl-2H-1,2,3,4-tetrazole
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
(3aR,6aS)-2-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
N-methyl-1-phenyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-cyclopropyl-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
2-{[4-(2-amino-1,3-benzothiazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
(2S,4R)-4-amino-1-(3-cyclopentaneamidobenzoyl)-N-methylpyrrolidine-2-carboxamide
1-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}azetidin-3-ol
3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-[(3-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-N-(3-methylphenyl)methanesulfonamide
3-(5-methyl-1H-pyrazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
2-(3-methyl-4-{[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
2-methoxy-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}pyrimidine-5-carboxamide
1-{4-[(butan-2-yl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[(3-fluorophenyl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide