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1-(6-methyl-2-propylpyrimidin-4-yl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-4-amine
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
7-[(2,3-difluorophenyl)methyl]-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
methyl 2-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]acetate
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]isoquinoline
3-(2H-1,3-benzodioxol-5-yl)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]propan-1-one
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2-hydroxyethyl)-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-benzyl-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-(4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
1-{4-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]benzoyl}piperidine
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
4-(4-chlorophenyl)-1-(thiomorpholin-4-yl)butan-1-one
3-(2-fluorophenyl)-1-[4-(furan-2-carbonyl)piperazin-1-yl]-3-phenylpropan-1-one
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-phenylacetamide
N-benzyl-2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}acetamide
6-[4-(cyclopropylmethyl)piperazin-1-yl]-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-(1-methyl-1H-indole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl 3-[2-(4-methylphenoxy)acetyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
1,3,5-trimethyl-4-({3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)-1H-pyrazole
6-[(3-aminopyrrolidin-1-yl)methyl]-N-(2H-1,3-benzodioxol-5-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
1-benzyl-N,N-dimethyl-5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzyl-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(4-ethylphenyl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl][(2-phenyl-1,3-thiazol-5-yl)methyl]amine
1-ethyl-N-[3-(2-fluorophenyl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
N,2-dimethyl-6-(2-methylpropyl)-N-[1-(pyridin-2-yl)ethyl]pyrimidine-4-carboxamide
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
5-[1-(but-2-ynoyl)piperidin-4-yl]-3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
1'-[3-(difluoromethoxy)benzoyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(hydroxymethyl)-4-({3-[2-(3-hydroxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-2-methylpyridin-3-ol
(1S,5R)-6-(cyclopropylmethyl)-3-(quinoxalin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-methoxy-3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indol-2-one
1-{1-[2-(1H-indol-3-yl)ethyl]piperidin-4-yl}pyrrolidin-2-one
3-{1-[2-(4-phenylphenyl)acetyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(benzyloxy)-8-[2-(thiophen-3-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
3-methyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)but-2-enamide
4-{4-[3-(4-methoxyphenyl)propanoyl]piperazin-1-yl}-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(3R,4S)-1-(1H-indazole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-4-methyl-1,4-diazepane
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
N-{[1-(dimethylsulfamoyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
3-[(dimethylamino)methyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-3-ol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-8-methoxy-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-methoxy-N-({5-[(1-methyl-1H-indol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide