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1-(2-{[(3-hydroxypiperidin-3-yl)methyl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpyridine
(3-ethyl-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methanol
5-[1-(2-fluorophenyl)cyclopropyl]-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
(1-methyl-1H-imidazol-2-yl)(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
1-[1-(3-cyclopentylpropyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
N-methyl-1-(oxan-4-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]piperidine-3-carboxamide
8-[2-(pyridin-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
7-fluoro-N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]quinoline-4-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-(5-fluoro-2-methylbenzenesulfonyl)piperidine
1'-[(4-chloro-2-fluorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(cyclohex-1-en-1-yl)-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-methanesulfonylbenzoyl)-3-(2-methoxyphenoxy)azetidine
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(3S,4R)-1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(6-methoxy-2,6-dimethylheptyl)-1-methyl-1H-1,3-benzodiazole
(1S,6R)-9-[2-(7-methoxy-4-methyl-2-oxo-2H-chromen-3-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[3,5-dimethyl-4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1H-pyrazol-1-yl]ethan-1-ol
4-methoxy-6-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
5-(2-cyclopropyl-1,3-benzoxazol-5-yl)-1,3,6-trimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-({1-[(4-methylphenyl)methyl]-5-oxopyrrolidin-3-yl}formamido)acetic acid
N-[2-({6-methylpyrazolo[1,5-a]pyrimidin-3-yl}formamido)ethyl]pyridine-3-carboxamide
3-methyl-7-[3-(pyridin-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}acetamide
2-(dimethylamino)-N-(3-hydroxypropyl)-2-(2-methylphenyl)acetamide
3-{1-[1-(2,6-dimethylphenoxy)propan-2-yl]-1H-imidazol-2-yl}pyridine
2-{[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
4-[6-(propan-2-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-methyl-N-[(6-methylpyridin-2-yl)methyl]-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
2-(4-{4-[(dimethylcarbamoyl)amino]phenyl}phenyl)-N,N-dimethylacetamide
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-4-yl)-decahydro-2,7-naphthyridin-2-yl]-2-cyclobutylethan-1-one
9-methyl-3-(2-methyl-1-benzofuran-7-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(prop-2-en-1-yloxy)phenyl]methyl})amine
2-hydroxy-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-(5-chloro-2-methoxyphenyl)-3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-4-yl)piperazine
1-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{[5-(4-methanesulfonylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}acetamide
(2S)-2-({[6-methyl-2-(prop-2-en-1-yloxy)quinolin-3-yl]methyl}amino)-3-phenylpropanamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
(1-{[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]methyl}cyclopropyl)methanol
5-(2,2-diphenylacetyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(oxan-4-yl)piperidine-3-carboxamide
3-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-6-methoxy-1H-indazole
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(hydroxymethyl)piperidin-3-ol
3,5-dichloro-N,4-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]benzamide