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N-(1-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-1-oxopentan-2-yl)acetamide
8-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[(2S)-pyrrolidin-2-ylmethyl]urea
[(2S,4R)-1-(3,5-dichloro-4-methylbenzoyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
N2-[1-(cyclohexylmethyl)piperidin-3-yl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl](pyridin-2-yl)methanol
1-(2,6-dimethylpyridin-4-yl)-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazine
1-(4-ethylpiperazin-1-yl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]propan-1-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-(3-chlorophenyl)-3-cyclopropyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazole
5-methyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-(2,6-dimethoxyphenyl)-4-phenyl-1H-imidazole
N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
7-chloro-2-[2-(propan-2-yl)pyrimidin-5-yl]-4-(pyrrolidine-1-carbonyl)quinoline
5-(4-methoxy-2-methylphenyl)-4-(4-methylphenyl)-2-(4-methylpiperazin-1-yl)pyrimidine
{[3-(cyclopentyloxy)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
[(2-chloro-4,5-dimethoxyphenyl)methyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1-(furan-2-ylmethyl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)piperidine-4-carboxamide
methyl 5-{[(6-methylpyridin-2-yl)methyl]amino}-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperidin-4-amine
(3R,4S)-4-[4-(4-cyclopentylpyrimidin-2-yl)-1,4-diazepan-1-yl]oxolan-3-ol
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-pyrazol-4-yl)benzamide
3-{[cyclopentyl(prop-2-en-1-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[(1-{6-[(2-cyclopentylethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-(azepan-1-yl)-3-[3-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-[(3S,4R)-1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
6-methyl-2-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)quinolin-4-ol
N2-(3,3-dimethylcyclohexyl)-N1-(pyridin-3-yl)ethane-1,2-diamine
methyl 6-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylate
7-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(1S,5R)-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
N-(5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}-4-methyl-1,3-thiazol-2-yl)acetamide
5-{[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2,1-benzoxazole
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-N-methylpyridin-2-amine
2-[benzyl(methyl)amino]-N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
{1-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(propan-2-yl)propanamide
5-(4-fluoro-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-methoxy-5-methyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
4-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-3-methyl-N-(propan-2-yl)benzamide
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-methylpyridine-3-carboxamide
4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-(4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine