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N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiophene-2-carboxamide
2-(3-ethoxyphenyl)-5-(methanesulfonylmethyl)pyridine
(4aS,8aR)-2-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-decahydroisoquinoline
N2-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-methylpyrimidine-2,4-diamine
2-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-[1-(4-methylphenyl)ethyl]acetamide
N-[3-(3-chlorophenyl)phenyl]-1-[(2-ethylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
2-(dimethylamino)-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylbenzamide
1-[(3-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-({7-[(2-butyl-1H-imidazol-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
N-{[1-(2-chloro-4-fluorobenzenesulfonyl)piperidin-3-yl]methyl}furan-2-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}){[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-{3-[cyclopentyl(methyl)amino]propyl}-5,6-dimethylpyrimidin-4-amine
1-(1-benzofuran-2-ylmethyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3S,4S)-1-(1-methyl-4-phenylpiperidine-4-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-benzyl-1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methylpiperidin-3-amine
N-[2-(2,3-dimethoxyphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-({2-[2-(4-fluorophenoxy)ethyl]phenyl}methyl)propanamide
3-(2-methylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
3-({1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl}methyl)-1-phenylurea
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)(oxan-4-ylmethyl)amine
4-{2-amino-3-cyano-8-hydroxy-5H,6H-benzo[h]quinolin-4-yl}benzamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
5-chloro-3-fluoro-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-(1-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-(2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}pyrimidin-4-yl)piperidin-3-ol
2-[4-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)-1H-pyrazol-1-yl]ethan-1-ol
N-{[2-(difluoromethoxy)phenyl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
3-[(3-fluorophenyl)methyl]-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
methyl 3-(2-methoxyacetamido)-1-(3-phenylpropyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]ethyl}-6-methyl-3,4-dihydropyrimidin-4-one
1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-(hydroxymethyl)phenol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-methyl-7-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N3-cycloheptyl-1-cyclopropyl-N5-[(2,3-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-(2,6-dimethylphenyl)urea
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-3-carboxamide
2-amino-6-cyclopropyl-4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}pyridine-3-carbonitrile
4-(8-hydroxyquinolin-2-yl)-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(2-oxopiperidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
2-methyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-(morpholin-4-ylmethyl)-1,4-oxazepane