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N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
(3R)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
1-(2-{[(3-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}ethyl)pyrrolidin-2-one
3-(4-fluorophenoxymethyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
2-(cyclopropylmethyl)-7-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}cyclobutanecarboxamide
5,6-dimethoxy-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2-dihydroisoquinolin-1-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-indol-3-yl)ethyl]benzamide
3-(2-phenylethyl)-8-(1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(pyrrolidin-1-ylmethyl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
2-[5-(5-methoxy-4-oxo-1,4-dihydropyridin-2-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]acetic acid
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]-6-methylphenol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methylpropanamide
1-{5-[(4-ethylpiperazin-1-yl)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
N,1,3-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(2-phenylethyl)piperidin-2-one
N-[1-(4-hydroxyphenyl)propyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
4-(1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)morpholine
2-(4-fluorophenyl)-N-[2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(2-fluorophenyl)methyl]-3-[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-3-yl]propanamide
2-[4-(4-{[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]-1-(pyrrolidin-1-yl)ethan-1-one
1-(4-ethyl-5-methylpyrimidin-2-yl)-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
1-(2-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
2-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}butanamide
1-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
8-(2,2-dimethylpropyl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-({1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzamide
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methylacetamide
N-cyclohexyl-N-(pyridin-2-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenyl)-3H,4H,5H,7H-thieno[3,4-d]pyrimidin-4-one
(3S,4S)-1-(4-chlorobenzoyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
6-chloro-2-(2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
(3R,4S)-1-[6-(methoxymethyl)pyridine-2-carbonyl]-4-propylpyrrolidin-3-amine
N-[3-(pyridin-2-yl)propyl]-4-(pyridin-4-yl)pyrimidin-2-amine
methyl 6-[(2E)-3-phenylprop-2-enoyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(piperidin-1-yl)-2-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
1-(2-ethoxyacetyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-4-carboxamide
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,7S)-5-[5-(ethylcarbamoyl)pyridin-2-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-[3-oxo-3-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)propyl]acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(2-methoxyethyl)-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid