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1-tert-butyl-N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(3R,7S,8aS)-7-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
4-(cyclopropylmethyl)-1-(5-fluoro-1H-indole-2-carbonyl)-1,4-diazepan-5-one
{1-[(2-aminopyridin-3-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-cyclopropyl-5-[(E)-2-phenylethenesulfonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
6-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,2-dimethylpropanamide
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)butan-1-one
ethyl 2-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]acetate
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
ethyl 1-{5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
1-{5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
3-(3-fluorophenyl)-4-[4-(2-oxopyrrolidin-1-yl)benzoyl]piperazin-2-one
3-acetyl-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-1H-pyrazole-5-carboxamide
N-{[5-(2-amino-6-methoxypyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
4'-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aS,6aS)-2-(2-chloro-6-fluorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(furan-2-yl)-1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]propan-1-one
6-ethoxy-3-{[methyl(propan-2-yl)amino]methyl}-1,2-dihydroquinolin-2-one
N-[2-methyl-5-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
3-(1-methylpiperidin-3-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]propanamide
(3R,4S)-N,N-dimethyl-4-(propan-2-yl)-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-amine
(5S,9aS,9bS)-5-(4-phenylphenyl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}propanamide
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
ethyl 5-[(4-hydroxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(oxolan-2-ylmethyl)-3-[2-(propan-2-yl)phenyl]-1-(pyridin-2-ylmethyl)urea
(3S,9aR)-8-(3-methoxybenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 5-(cyclohexylamino)-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-[5-(4-chlorophenoxy)-1,3-dimethyl-1H-pyrazol-4-yl]-7-hydroxy-1,2,3,4-tetrahydroquinolin-2-one
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
5-cyclopropyl-3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1,2,4-oxadiazole
(4aR,7aS)-1-(cyclopropylmethyl)-4-(morpholine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopentyl-N-({4-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)naphthalene-1-carboxamide
N-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(quinolin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
N-methyl-2-{4-[({[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}carbamoyl)amino]phenyl}acetamide
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-3-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
N-(1-carbamoylcyclopentyl)-4-[(3-hydroxypiperidin-1-yl)sulfonyl]benzamide
(3R,4S)-4-(3-methoxyphenyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine