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N-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
3,5-dichloro-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-4-(prop-2-en-1-yloxy)benzamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
4-[3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]-2-[(3,4,5-trimethoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-ol
2-methoxy-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyridine-3-carboxamide
(2R,6R)-1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-oxo-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholine-2-carboxamide
2-methyl-6-[1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidin-4-yl]pyrimidin-4-ol
1-cyclopropyl-N-[(5-fluoro-2-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,3-dimethyl-1H-indole-2-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-(2,5-dihydro-1H-pyrrole-1-carbonyl)piperidine
2-({4-[5-(2-fluorophenyl)furan-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-imidazole
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
4-(1H-imidazol-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
(1S,3R)-3-amino-N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]cyclopentane-1-carboxamide
1-{[(2-fluorophenyl)methyl]carbamoyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3aR,7aS)-2-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
4-benzyl-1-(cyclobutylmethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methoxyethyl)-8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
7-(2-methoxyethyl)-2-{[4-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
methyl 5-[1-(carbamoylmethyl)piperidine-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2,3-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-indole-5-carboxamide
methyl (2S)-1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
2-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N,N-dimethylpyridine-3-carboxamide
6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,3-dihydropyridazin-3-one
2-cyclopentyl-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}acetamide
3-methoxy-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
2-methoxy-N-[(3R,4S)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-methyl-2-{2-[methyl(oxan-4-ylmethyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N,N,2,2,3-pentamethylcyclopentane-1-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-cyclopropylpyrimidin-4-amine
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-methyl-8-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
5-acetyl-N-[(5-ethylpyridin-2-yl)methyl]-N-methylthiophene-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[2-(2,3-dichlorophenyl)ethyl]-1-methylazepane-2-carboxamide
3-fluoro-5-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]acetamide
N-methyl-3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-[2-(methylsulfanyl)ethyl]benzamide