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N-(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}piperidin-4-yl)methanesulfonamide
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-fluoro-N-methyl-2-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(methoxymethyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
7-(cyclohexylmethyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)urea
N6-cyclopropyl-N4-methyl-N4-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4,6-triamine
4-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]benzamide
1-methyl-4-phenyl-3-[1-(9H-purin-6-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[(dimethylcarbamoyl)(phenyl)methyl]-N'-(4-methylphenyl)propanediamide
5-ethyl-1'-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(diethylamino)-3-[5-({[(2,6-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-propyl-1H-pyrazole-5-carboxamide
4-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(2-fluorophenyl)-N-(oxan-2-ylmethyl)propanamide
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}[(5-methylthiophen-2-yl)methyl]amine
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyrimidin-2-amine
N,N-dimethyl-3-[1-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-3-yl]propanamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
6-phenyl-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]pyridine-3-carboxylic acid
3-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrol-3a-ylformamido]-N-(2,5-difluorophenyl)propanamide
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2-methylphenol
N-{2-[(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}methanesulfonamide
N-[3-(pyridin-4-yl)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-4-ylmethyl)piperidine
1-benzyl-N3-ethyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(furan-2-carbonyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-(3-methylbut-2-en-1-yl)-8-(thiophene-2-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
4-(hydroxymethyl)-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
4-cyclopentanecarbonyl-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
methyl 2-({[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)acetate
N-[1-(methoxymethyl)cyclopentyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-(azocan-1-yl)-1-[4-(1-methoxypropan-2-yl)piperidin-1-yl]propan-1-one
1-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-N-(3-hydroxypropyl)piperidine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]pyridazine-4-carboxamide
4-methyl-N-(3-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)benzamide
3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2,6-dimethylpyrimidine-4-carboxamide
1-{1-[2-(3-fluoro-4-hydroxyphenyl)acetyl]piperidin-3-yl}-3-phenylpropan-1-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
(1S,5R)-3-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(dicyclopropylmethyl)methylamine
3-cyclohexyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-2,1,3-benzothiadiazole