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3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-cyclohexyl-3-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}propanamide
1-acetyl-N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]piperidine-4-carboxamide
3-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}pyrrolidin-2-one
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-{[5-(1-cycloheptylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
2-(1H-pyrazol-1-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-(4-benzyl-1H-pyrazol-5-yl)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
3,3-dimethyl-1-({5-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
3-methyl-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}urea
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,2-dihydroisoquinolin-1-one
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
5-[(2-cyclohexylpyrimidin-5-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(2-hydroxyethyl)-4-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}sulfamoyl)benzamide
4-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}thiomorpholine
2-methyl-4-(propan-2-yl)-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
3-(4-fluoro-3-methylphenyl)-1-methyl-6-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-4-ol
1-cyclopropanecarbonyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-4-carboxamide
4-cyano-N-(2-fluoro-4-methoxyphenyl)-4-phenylpiperidine-1-carboxamide
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-cyclopropyl-1-{[(2-phenylethyl)carbamoyl]methyl}pyrrolidine-3-carboxylic acid
3-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-[2-(piperidin-1-ylmethyl)phenyl]urea
2-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(3-methoxybenzoyl)piperazine
1-(2-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
1-{2-[ethyl(methyl)amino]acetyl}-4-(2-methylphenoxy)piperidine-4-carboxylic acid
8-cyclopropanecarbonyl-2-(1-methyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(6-methoxypyridin-3-yl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}morpholine
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
1-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[2-(pyridin-4-yl)ethyl]piperidin-4-amine
1-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
(2S,4S)-1-(2-ethoxyethyl)-N-ethyl-4-(2-hydroxy-4-methylbenzamido)pyrrolidine-2-carboxamide
(2S,4S)-N,N-diethyl-1-(naphthalen-2-ylmethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-cyclohexyl-1-(2-ethoxyethyl)-2-oxo-N-propyl-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[(2,6-difluoro-4-methoxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
4-(2-ethylpyrimidine-5-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
[(4-fluorophenyl)methyl](1H-indol-5-ylmethyl)(pyridin-4-ylmethyl)amine
4-[4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
(1S,5R)-6-[(2-chloro-5-fluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(adamantan-1-yl)-4-hydroxy-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide