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4-methyl-3-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,4-dihydroquinoxaline-2-carboxamide
1-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
5-fluoro-2-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
4-(1-methyl-1H-pyrazole-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
7-(3-chlorophenyl)-4-(furan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2,2-dimethylpropan-1-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,3-thiazole-4-carboxamide
7-fluoro-3-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-1,2-dihydroquinolin-2-one
N-[3-(cyclohexyloxy)propyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
1-[(3-methylphenyl)methyl]-4-(pyrrolidine-3-carbonyl)piperazine
(3S,4R)-1-{3-[4-(dimethylamino)phenyl]propanoyl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
5-[(3-ethoxypropyl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
{2-methyl-6-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyrimidin-4-yl}methanamine
N-methyl-2-(1H-pyrazole-3-carbonyl)-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-amino-3,5-dibromobenzene-1-sulfonamide
(2S,3R)-2-methylmorpholine-3-carboxylic acid
2-[(3-fluorophenyl)methoxy]-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
(2R)-2-amino-3-carbamoylpropanoic acid hydrate
(2R)-2-amino-3-[(2-methylbutan-2-yl)sulfanyl]propanoic acid
(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-(3,4,5-trifluorophenyl)propanoic acid
tert-butyl 2,5-diaminopentanoate hydrochloride
4-chloro-2-[(cyclopentylmethyl)sulfanyl]pyridine
5-nitro-3-[4-(trifluoromethyl)phenyl]-1H-indazole
5-bromo-2-methanesulfinylpyrimidine
5-ethylpyrimidin-4-ol
(2S)-2-acetamido-4-methylpentanoic acid
4-{[(4-fluorophenyl)imino]methyl}phenol
[6-(trifluoromethyl)pyrimidin-4-yl]methanol
4-bromo-2-(tert-butoxy)pyridine
(3S)-1-methylpiperidin-3-amine
tert-butyl N-[(1S)-3-hydroxy-1-phenylpropyl]carbamate
3-phenylpyridine-4-carboxylic acid
4,5-dichloro-2,3-dihydro-1H-isoindol-1-one
penta-2,4-dienoic acid
3-(3-bromopyridin-2-yl)-3,9-diazaspiro[5.5]undecane
4-(3-carboxyphenyl)-2-chlorobenzoic acid
2-(pentan-3-yloxy)-4-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine
2,3-bis(chloromethyl)-6-(trifluoromethyl)pyridine
(2S)-2-methylpyrrolidine
3,4-dichloro-5-(3-methylbutoxy)pyridazine
(2R)-2-cyclohexyl-2-hydroxy-2-phenylacetic acid
1-(5-methylfuran-2-yl)propan-1-one
4-[6-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-yl]morpholine
rel-(3R,5S)-piperidine-3,5-dicarboxylic acid
[5-(6-bromopyridin-2-yl)pyridin-3-yl]methanol
1-[amino(phenyl)methyl]cyclopropan-1-ol
(1R)-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid