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3-(3-chlorobenzoyl)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
1-{imidazo[1,2-a]pyridine-6-carbonyl}-3-(thiophene-2-carbonyl)piperidine
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(5-methyl-1,3-benzoxazol-2-yl)pyrrolidin-3-yl]methanol
4-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
4-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
(4S)-3-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
(2S,4S)-4-amino-1-[(2-methoxypyridin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
2-methoxy-N-(2-methoxy-2-methylpropyl)-4-methylbenzamide
3-{4-[3-(pyrrolidin-1-yl)pyrazin-2-yl]phenyl}propanoic acid
1-(pyridin-3-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethane-1,2-dione
N-[2-(4-hydroxyphenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl 3-{[3-(methylcarbamoyl)-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}imidazolidin-2-one
1-(4-methoxyphenyl)-3-methyl-4-[(4-methylpiperidin-1-yl)sulfonyl]piperazin-2-one
4-{4-[3-(1-methylpiperidin-3-yl)propanoyl]piperazin-1-yl}benzonitrile
2-benzyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
3-cyclopropyl-5-(methanesulfonylmethyl)-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-N-methyl-1H-indole-2-carboxamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-{3-[3-(3-cyanopyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-phenylacetamide
N-(adamantan-1-yl)-5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
1-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N5-(1,4-dithiepan-6-yl)-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-{1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-cyclopropyl-1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
1-ethyl-6-{[4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-1H-indole
7-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
2-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}benzoic acid
2-(dimethylamino)-N-[3-({[(3-hydroxypiperidin-3-yl)methyl]carbamoyl}amino)-2-methylphenyl]acetamide
2,3-dimethyl-7-(piperidine-1-sulfonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-[1-(2,3-difluoro-6-methoxybenzoyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
2-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(morpholin-4-yl)-3-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-yl)propan-1-one
5-chloro-N-ethyl-N-(2-methoxyethyl)-3-phenyl-1H-indole-2-carboxamide
3-methyl-1-(4-{[1-(4-methylphenyl)propan-2-yl]amino}piperidin-1-yl)butan-1-one
3-[(2,3-dichlorophenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,3R)-2-amino-3-hydroxy-N-{[4-(methylsulfanyl)phenyl]methyl}-N-propylbutanamide
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2,4-difluorophenoxy)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[3-(dimethylamino)benzoyl]-1-(4-methylphenyl)piperazin-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
benzyl(methyl)[2-(morpholin-4-yl)propyl]amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-N-[(4-methylphenyl)methyl]-1H-imidazole-5-carboxamide