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1-({5-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
5-chloro-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]piperidine-3,4-diol
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2,5-dimethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-{4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
1-(2-phenoxyethyl)-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
5-(4-acetylphenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,2-oxazole-3-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-5-{[2-(5-methylfuran-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 2-(piperidine-1-sulfonyl)-6-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-cyclopentyl-3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}piperazin-2-one
ethyl 1-[(2-hydroxy-6-methoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(3S,4R)-1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
(4aS,8aS)-2-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-decahydroisoquinolin-4a-ol
4-{2-[1-(3-chloro-5-methoxybenzoyl)piperidin-2-yl]ethyl}morpholine
1-(pyrrolidin-1-yl)-3-[1-(quinolin-4-ylmethyl)piperidin-3-yl]propan-1-one
1-{4-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
N-(2-hydroxy-2-phenylethyl)-N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-benzyl-8-(5-fluoropentyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopropanecarbonyl-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-4-carboxamide
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-{[benzyl(methyl)amino]methyl}-N-(1H-imidazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
7-fluoro-3-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{1-[4-(3-chlorophenyl)-5-[(cyclohexylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpropanamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[(5-chloro-2-methoxyphenyl)methyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
1,2-dimethyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
N-(2-methyl-1,3-benzothiazol-6-yl)-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
1-cyclopentyl-N-methyl-5-oxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)pyrrolidine-3-carboxamide
(1H-imidazol-2-ylmethyl)({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
1-{[1-(quinolin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
methyl 4-[5-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(2-{2-[1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}propane-1-sulfonamide
N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)-2-(pyrrolidin-1-yl)propanamide
N-benzyl-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-4-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[1-(piperidin-1-yl)cyclohexyl]methyl}amine
1-[1-(2,3-dimethylphenyl)piperidin-4-yl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}acetamide
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
(2S,4S)-N-ethyl-4-[(1r,4r)-4-methylcyclohexaneamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
(4aS,8aR)-6-[(2-ethylpyrimidin-5-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(2,6-dimethoxybenzoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
5-(hydroxymethyl)-2-methyl-4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]pyridin-3-ol
4-(3,6-dimethylpyrazin-2-yl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperazine-1-carboxamide
1-(adamantan-1-yl)-4-(1,2-oxazole-3-carbonyl)piperazine