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7-(2,3-dimethoxyphenyl)-9-methoxy-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(isoquinolin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[(2-chlorophenyl)methyl](methyl)amino}-2-[4-(dimethylcarbamoyl)phenyl]acetic acid
{4-[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
1-(2-methoxyethyl)-5-{1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}piperidin-2-one
3-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-1-[2-(2-ethoxyethoxy)phenyl]urea
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-methyl-1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
1-(1H-imidazole-2-carbonyl)-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepane-6-carboxylic acid
3-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
ethyl 3-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)butanoate
2-(2,3-dimethoxyphenyl)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
N-[1-(1H-indol-1-yl)propan-2-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethoxy)ethan-1-ol
(4aS,8aR)-6-(1,3-dimethyl-1H-indole-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-methyl-N-[3-({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propyl]benzene-1-sulfonamide
1-cyclopentyl-N5-[2-(2-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4,6-dimethyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(thiophene-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-6-methoxypyrimidin-2-amine
3-oxo-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-2,3-dihydro-1H-indene-1-carboxamide
4-(ethanesulfonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
N-[3-(4-hydroxyphenyl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
ethyl 3-{[1-(cyclohexylmethyl)-3-(dimethylcarbamoyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
8-(3,6-dimethyl-1-benzofuran-2-carbonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
(2S,4S)-1-[(3-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(4aR,8aS)-6-[2-(4-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-3-(4-methylphenyl)propan-1-one
N-[1-(3-phenylpropyl)piperidin-3-yl]-4-(trifluoromethyl)pyrimidin-2-amine
5-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 2-(benzylsulfamoyl)-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-fluoro-2-hydroxybenzoyl)-4-(hydroxymethyl)azepan-4-ol
4-[(4-methyl-5-{1-[(3-methylphenyl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
13-[4-(dimethylamino)phenyl]-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
5-(2-fluoro-4-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-(4-methylpiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
1-(1-methoxybutan-2-yl)-4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
1-methyl-3-[1-(2-oxo-1,3-oxazolidine-4-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-methylpyrazin-2-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
5-chloro-N,4,6-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 2-{methyl[1-(pyridin-4-yl)ethyl]carbamoyl}acetate
1-(3-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}pyridine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-2-yl)acetamide