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2-{5-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-(2-methylphenyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-diazepane
4-methyl-5-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1,2,3-thiadiazole
2-[(3R,4R)-3-hydroxy-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl]pyridine-4-carboxamide
2-(cyclopropylmethyl)-8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-(4-fluorophenyl)piperidine
2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1H-indole-3-carboxamide
1-cyclohexyl-N3-cyclopropyl-N5-[(3-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3R,4S)-1-[2-(3,4-dimethylphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]propanamide
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1,3-dimethylpiperazin-2-one
6-ethyl-5-methyl-N4-{[4-(piperidine-1-carbonyl)phenyl]methyl}pyrimidine-2,4-diamine
2-[3-(furan-2-yl)-5-(5-methoxy-1,2-dimethyl-1H-indol-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
(4aR,8aS)-1-[3-(1H-imidazol-1-yl)propyl]-6-(2-methylpropanoyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
4-fluoro-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
2-methoxy-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
(1S,5R)-6-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(2-methylphenyl)ethan-1-one
3-{[1-(3-fluoro-2-methoxybenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
2-methyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-phenoxyethan-1-one
N-(1-{1-[(4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(3aR,6aR)-2-(oxane-4-carbonyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1,3-benzoxazol-2-yl)-N-[2-(2-methoxyphenoxy)ethyl]piperidin-4-amine
1-cyclohexyl-5-(furan-2-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(5-{[2-(furan-2-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
2-({[(3R,4R)-4-(hydroxymethyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
[({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)sulfamoyl](ethyl)methylamine
ethyl 4-{3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazine-1-carboxylate
8-(5-methylpyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 2-[3-(2-{[(5-methylfuran-2-yl)methyl]carbamoyl}ethyl)piperidin-1-yl]pyridine-3-carboxylate
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-(dimethylsulfamoyl)-N-[(2-methoxyphenyl)methyl]morpholine-2-carboxamide
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}morpholine-2-carboxylic acid
4-(2-methoxy-5-methylphenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
(1S,5R)-3-(oxan-4-yl)-6-(1-phenyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,3S,5S)-8-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
3-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}-1λ6-thiolane-1,1-dione
N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-ethyl-9-[2-(propan-2-yl)pyrimidin-4-yl]-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
1-(2-methyl-5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
9-[(4-fluoro-2-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}oxan-4-amine
5-(4-methyl-2-phenylpiperazine-1-carbonyl)-N-phenylpyrimidin-2-amine
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[(2-methylphenyl)(thiophen-2-yl)methyl]acetamide
1-(propan-2-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}piperidine-4-carboxamide
5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-propylpyrimidine