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2-{[4-(3-methoxypyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-(3-methoxypropyl)-6-[2-(pyridin-2-yl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{[4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
2-propyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,3-thiazole-4-carboxamide
2-(3-hydroxyadamantan-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
2-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethoxy)ethan-1-ol
6-(methoxymethyl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]pyrimidin-4-amine
7-chloro-3-({methyl[(1-methylpyrrolidin-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(pyridin-3-yl)piperidin-4-ol
3-[({1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
2-(1-benzyl-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl)ethan-1-ol
2-methyl-5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-[5-(2,6-dimethylpyrimidin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridin-3-amine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}acetic acid
4-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-N-(pyridin-3-yl)benzamide
1-cyclopropyl-5-oxo-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
4-[1-(methoxymethyl)cyclopropanecarbonyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl (2S,4S,5R)-1,2-dimethyl-4-{[2-(3-methyl-1H-pyrazol-1-yl)ethyl]carbamoyl}-5-(2-methylphenyl)pyrrolidine-2-carboxylate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl})amine
N-benzyl-5-[(4-acetamidophenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-fluoro-2-methoxybenzamide
(3S,4R)-1-[(4-methanesulfonylphenyl)methyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
5-cyclobutanecarbonyl-1'-(morpholine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(5-methyl-4-phenylthiophene-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(propan-2-yl)-3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
(2S,4S)-4-cyclobutaneamido-N-ethyl-1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidine-2-carboxamide
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[benzyl(methyl)amino]-3-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidine-3-carboxamide
1-[3-(furan-2-yl)propanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-{[6-(3-chlorophenyl)-7-(cyclopropylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
(3S)-1-(1-methyl-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-2-yl)pyrrolidin-3-ol
(4aS,8aR)-1-(3-aminopropyl)-6-(1-phenylcyclopropanecarbonyl)-decahydro-1,6-naphthyridin-2-one
2-methyl-4-{5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}but-3-yn-2-ol
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)but-3-enamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
4-{4-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-1-yl}phenol
(2R,3R)-3-{[(2,6-difluoro-3-methoxyphenyl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]benzonitrile
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-1-(2-methylphenyl)piperazin-2-one
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
1-(3-benzoylpiperidin-1-yl)-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(methoxymethyl)furan-2-carboxamide