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3-methyl-8-(thiophen-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
4-[(3-methoxyphenyl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
3-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-(2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
1-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
3-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-methyl-3-phenyl-8-[(1-propyl-1H-imidazol-2-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1S,6R)-9-(2,2-diphenylacetyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-amino-4-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-thiazole-5-carboxamide
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
4-ethanesulfonamido-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]benzamide
2-(dimethylamino)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(4-methylphenyl)acetamide
3-{[(1-benzothiophen-5-ylmethyl)amino]methyl}-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
2-phenyl-N-[2-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-methyl-4-{3-[4-(pyridin-4-yl)-1,4-diazepane-1-carbonyl]phenyl}butan-2-ol
2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
(1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carbonyl}piperidin-4-yl)methanol
3-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-5-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]benzamide
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
1-(2-aminoethyl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-{3-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-N-[2-(naphthalen-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-(1-benzofuran-2-yl)-1-[1-(4-methanesulfonylphenyl)ethyl]-1H-imidazole
4-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})(pyridin-3-ylmethyl)amine
[(3R,4R)-1-(2-methoxy-6-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-2-(propan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(morpholin-4-yl)propanamide
6-methyl-2-{[2-(pyridin-3-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
1-benzyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-pyrazole-4-carboxamide
methyl 4-{[2-oxo-5-(3-phenylpiperidin-1-yl)azepan-1-yl]methyl}benzoate
11-(3-chloro-5-methoxybenzoyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
4-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-[2-(2-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl})amine
3-chloro-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]thiophene-2-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]pyridazine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3,6-dimethyl-1-benzofuran-2-carboxamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
1-ethyl-N-methyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
(1S,5R)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(3-hydroxy-4-methylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one