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1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)pyrrolidin-3-amine
methyl 5-[4-(3-fluorophenoxy)piperidin-1-yl]-5-oxopentanoate
4-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1'-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
8-(2-methyl-2-phenoxypropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-oxo-N-[(2-phenoxypyridin-3-yl)methyl]pyrrolidine-3-carboxamide
1-({[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}methyl)piperidine-4-carboxamide
2-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-5-methoxyphenol
2-(3-{[methyl(oxan-4-ylmethyl)amino]methyl}phenyl)-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
(3R,4S)-4-(4-{[3-(2-hydroxyethoxy)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
1-cyclopropyl-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}acetamide
[4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-1,4-oxazepan-6-yl]methanol
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-(2-oxopyrrolidin-1-yl)acetamide
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-methyl-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
(3S,4R)-1-[2-(4-fluorophenyl)acetyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-propyl-N-(pyrrolidin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-ethylpiperidine-3-carboxamide
2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
3-(1-ethyl-1H-imidazol-2-yl)-1-(1H-pyrrole-3-carbonyl)piperidine
(2S,4S)-4-amino-1-(1-benzothiophene-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(2-benzylmorpholin-4-yl)pyridine-3-carboxamide
N-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,3-dimethylcyclohexan-1-amine
1-({6-[methyl(2-phenylethyl)carbamoyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-4-carboxamide
2-amino-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
[3-benzoyl-9-(2-methoxyethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
3-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
2-{1-methyl-4-[(1-methyl-1H-1,2,3-benzotriazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
5-[2-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidin-1-yl)-2-oxoethyl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
(3R,4R)-4-cyclopropyl-1-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
4-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}-2-ethylpyrimidine
N-[(2R,3R)-2-ethoxy-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-methyl-4-{3-methyl-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}piperidine
2-methyl-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1,8-naphthyridine-3-carboxamide
1-(3-methoxypyrazin-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{2-[methyl(phenyl)amino]acetyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[(2-chlorophenyl)methyl]-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
3-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl](pentan-3-yl)amine
2-methoxy-1-(4-{4-[3-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[6-(dimethylamino)pyridin-3-yl]pyridine-3-carbonitrile
1-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
N-({8-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
3-{2-oxo-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2-chlorophenoxy)ethan-1-one