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N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-4H-1,2,4-triazole
5-(2-chloro-4-methoxyphenoxymethyl)-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-pyrazole
7-(5-chloropyridin-2-yl)-4-(1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(5-{[(oxolan-2-ylmethyl)carbamoyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-ethyl-2-[1-(furan-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]pyridine
N-methyl-1-(2-phenylethyl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
(1R,5S,6R)-N-(furan-2-ylmethyl)-3-[(2-hydroxy-3,5-dimethylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[methyl(quinolin-5-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
4-(pyridin-2-yl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-ol
methyl 2-[1-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)-3-oxopiperazin-2-yl]acetate
{[6-(isoquinolin-5-yl)pyridin-3-yl]methyl}dimethylamine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-imidazol-1-yl)propyl]amine
N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-propylbenzoyl)piperidin-3-yl]propan-1-ol
1-{6-[4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3,4-difluorophenyl)propan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-(2-methyl-1-benzofuran-7-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(methoxymethyl)-1-[2-(4-methoxyphenoxy)ethyl]piperidine
(3aS,6aR)-5-(2-methylfuran-3-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[2-(azepan-1-yl)-2-oxoethyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[4-(4-chlorophenyl)butanoyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-ethyl-8-(9H-purin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(4-hydroxyphenyl)benzamide
[5-({8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decan-1-yl}methyl)furan-2-yl]methanol
9-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[1-(hydroxymethyl)cyclobutyl]methyl}-1-(2-methoxy-5-phenylphenyl)-3-methylurea
4-[(2-amino-5-methylpyrimidin-4-yl)amino]-1-(2-methoxyethyl)pyrrolidin-2-one
1-(3-chloro-4-methylphenyl)-3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-(3-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)azepane
1-{2-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
methyl 3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]benzoate
1,7-dimethyl-5-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
(2S,4S)-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-ethyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(butan-2-yl)(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-2-{4-phenyl-5-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-1-yl}butanamide
4'-[(2,3-dimethoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(5,6-dimethylpyrimidin-4-yl)-N-methylpiperidin-3-amine
3-(oxolan-3-yl)-5-[5-(propan-2-yl)thiophen-3-yl]-1,2,4-oxadiazole
(1S,5R)-6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(oxolane-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-(1-cycloheptylpiperidin-3-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(2-methyl-1H-imidazol-1-yl)butanamide
3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
(3S,4R)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-methyl-3-(2-methylpropyl)piperidin-4-ol