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2-[3-methyl-4-({methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
dimethyl(3-{2-[1-(4-methylquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
4-[3-(1H-1,2,4-triazol-3-yl)benzoyl]morpholine
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2,4-dimethylpyrimidine-5-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,N-dimethyl-4-[(3-methyl-1-benzofuran-2-yl)methyl]piperazine-1-sulfonamide
2-ethyl-5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
1-{3-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-indazole
N-(3-{4-[(9H-fluoren-9-yl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
(2R,3R,6R)-5-[(2,5-difluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
6-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
5-acetyl-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1S,5R)-3-[3-(1H-imidazol-2-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(morpholine-4-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
7-(5-chloropyridin-2-yl)-4-(3-methoxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-2-carbonitrile
(1S,6R)-9-(3-methylfuran-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
5-[4-(adamantan-2-yl)piperazin-1-yl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-(3-cyano-4-methoxyphenyl)-4-(pyridin-4-yl)piperidine-1-carboxamide
(2S)-1-acetyl-N-(furan-2-ylmethyl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
3-chloro-6-[4-(2-methoxyphenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
methyl(quinolin-6-ylmethyl)[(4-{2-[4-(thiophene-2-sulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
N-(3-benzamido-4-methoxyphenyl)-1H-imidazole-5-carboxamide
1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1H-indole
1-{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(1S,5R)-N-(3-chloro-4-fluorophenyl)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(2-methylquinolin-4-yl)-4H-chromen-4-one
2-{4-[(4-methyl-3-oxopiperazin-1-yl)methyl]phenyl}-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
1-{2-[1-(dimethylsulfamoyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
7-(3-chlorophenyl)-4-[(2-ethylpyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)propan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(4-methoxyphenyl)cyclopropyl]formamido}acetic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine-3-carboxylate
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
2-[1-butyl-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
(3S,4R)-4-(2-methylphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidine-3-carboxylic acid
1-ethyl-N-(1-hydroxybutan-2-yl)-3-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
(3R,4S)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-amine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1-methylcyclopropanecarbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3-ethylphenyl)-3-[(1-methanesulfonylpiperidin-4-yl)amino]propanamide
1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-cyclopropyl-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
(1S,4S)-2-(2-chlorophenyl)-5-[2-(naphthalen-1-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one