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N-methyl-N-(1,3-thiazol-2-ylmethyl)-2-{4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]morpholin-3-yl}acetamide
(4aS,8aR)-6-(1-aminocyclobutanecarbonyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
8-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decan-3-ol
2-{5-[4-(hydroxymethyl)phenyl]-1H-indol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-ethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(benzyloxy)-1-[2-(4-methylpiperazine-1-carbonyl)piperazin-1-yl]ethan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(1,3-thiazole-4-carbonyl)piperidin-3-amine
5-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-2H-pyran-2-one
2-(3-chlorophenyl)-N-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]acetamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(2,2,2-trifluoroethyl)-1H-1,3-benzodiazole-5-carboxamide
5-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-4-phenyl-1H-imidazole
1-[4-(3-chloropyridin-2-yl)piperazin-1-yl]-4-(piperidin-1-yl)butan-1-one
N-[(3S,4R)-1-[2-(benzyloxy)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-[(3-fluoro-2-methoxyphenyl)methyl]-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
N-[3-(4-ethylpiperazin-1-yl)propyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
methyl (2S)-1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxylate
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-methoxy-1-methyl-1H-indole-2-carboxamide
3-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-1-methyl-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
3-[(3R,4S)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-{2-ethyl-4-[3-(methoxymethyl)pyrrolidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}acetic acid
3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
N-cyclopentyl-4-(6-methylpyridazin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-3-[3-({methyl[1-(pyridin-3-yl)propyl]carbamoyl}amino)phenyl]propanamide
8-butanoyl-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-({[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
6-(methylsulfanyl)-2-(3-propyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
5-ethyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
(1R,7S)-3-(2,2-dimethylpropyl)-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
methyl 4-[(3-{[4-(1H-pyrazol-5-yl)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
2-(6-methoxynaphthalen-2-yl)-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
2-{5-[3-(3-methylbutanoyl)piperidine-1-carbonyl]pyridin-2-yl}benzoic acid
1-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}pyrrolidin-2-one
N-(6-fluoropyridin-3-yl)-2-(hydroxymethyl)piperidine-1-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(1H-1,2,4-triazol-3-yl)benzamide
3-{[(4-fluoro-2-hydroxyphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(3-chlorophenyl)-4-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propyl)piperazine
3-(2-methylpropyl)-5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazole
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(4-fluorophenyl)methyl]-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
5-[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]pyridine-2-carbonitrile
3-(azepane-1-carbonyl)-1-ethyl-N-[3-(pyridin-4-yl)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-2-(phenylsulfanyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-(2-phenylethyl)-6-[2-(trifluoromethyl)benzenesulfonyl]-6-azaspiro[2.5]octane-1-carboxamide
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one