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butyl({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-butyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
1-ethyl-N-methyl-6-oxo-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
4-(5-tert-butyl-1H-pyrazol-3-yl)-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(benzyloxy)methyl]-1-[(1R,2S)-2-phenylcyclopropyl]-1H-1,2,3-triazole
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
4-({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)-1λ6-thiomorpholine-1,1-dione
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)thiophene-2-carboxamide
N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
2-({[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-propyl-3-(pyridin-3-ylmethyl)urea
N-[2-(2,4-dichlorophenyl)ethyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-cyclopropyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}pyridine-2-carboxamide
2-[4-(3-chloro-2-fluorophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
8-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]quinoline
2-(2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-1,3-benzodiazole
6-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
8-fluoro-3-(1-methyl-5-oxopyrrolidin-3-yl)-3,4-dihydroquinazolin-4-one
N-(2,3-dihydro-1H-inden-2-yl)-5-(morpholin-4-ylmethyl)-N-propylfuran-3-carboxamide
N-[(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]naphthalene-1-carboxamide
3-[2-(furan-2-yl)-2-hydroxyethyl]-1-[4-(morpholine-4-carbonyl)phenyl]urea
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-2-yl]ethyl}phenol
(1R,4S)-1,7,7-trimethyl-N-[(5-methylthiophen-2-yl)methyl]-3-oxo-N-(prop-2-en-1-yl)-2-oxabicyclo[2.2.1]heptane-4-carboxamide
1-(azocan-1-yl)-3-(2-methoxy-4-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propan-2-ol
1-[2-(furan-2-yl)ethyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
2-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]-1,3-oxazole-4-carboxylic acid
ethyl 3-benzyl-1-[(2-chlorophenyl)carbamoyl]piperidine-3-carboxylate
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N,N-diethyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-[2-(3-methoxypyrazin-2-yl)phenyl]-1,3-benzoxazole
4-(1-{[ethyl(methyl)carbamoyl]methyl}piperidin-3-yl)benzoic acid
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
5-(methoxymethyl)-N-[2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(1,3-benzoxazol-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-(3-hydroxy-3-methylbutyl)-N-(2-hydroxybutyl)benzamide
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2-methylphenol
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-(morpholin-4-yl)butanamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-(methylsulfanyl)pyrimidine
2-(2-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-[2-(4-chlorophenoxy)ethyl]-3-methoxypiperidine
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)piperidin-3-amine
4-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyridazine
1-(2H-1,3-benzodioxol-5-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole