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5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
(3S,4S)-1-(3-cyclopentylpropanoyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
4-{[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]methyl}-1H-pyrazole-3-carboxylic acid
1-methyl-4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-[2-(4-hydroxypiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
(2S)-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}-2-phenylacetamide
2-(4-chloro-2-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
6-ethyl-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({2-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(4aR,8aR)-4a-hydroxy-7-[(2,4,5-trimethylphenyl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
1-methyl-9-[2-(phenylsulfanyl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-3-methoxypiperidine
(1S,5R)-3-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N'-[furan-2-yl(phenyl)methyl]-N-[2-(methylsulfanyl)phenyl]butanediamide
N-[(5-methylfuran-2-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyridine-3-carboxamide
4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
2'-amino-4'-(2-ethylpyrimidin-5-yl)-7',8'-dihydro-5'H-spiro[piperidine-4,6'-quinoline]-3'-carbonitrile
N-{[1-(3-chlorophenyl)pyrrolidin-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(2,6-dimethoxy-4-methylphenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
2-{2-[1-(furan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-pyrrol-1-yl}pyrimidine
N-[4-(difluoromethoxy)-2-methylphenyl]-4-(1-methylpiperidin-4-yl)piperazine-1-carboxamide
2-[2-(morpholin-2-yl)acetamido]-N-(pyridin-2-ylmethyl)benzamide
[(3R,4R)-1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carbonitrile
1-[2-(4-methoxyphenyl)ethyl]-N-[(5-methylfuran-2-yl)methyl]-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(3-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}phenyl)acetamide
4-[(4aS,8aR)-decahydroisoquinolin-2-yl]-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
5-ethyl-4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2,6-dimethylpyrimidine
4-{1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-2,1,3-benzoxadiazole
N-methyl-3-(2-methylpropyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
2-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}furan-2-yl)benzonitrile
(3S)-3-ethyl-4-[2-(3-methylphenyl)benzoyl]morpholine
1-[(3-fluorophenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
2-[5-(methylcarbamoyl)thiophen-2-yl]-N-[3-(methylsulfanyl)phenyl]pyrrolidine-1-carboxamide
3-[(4-fluorophenyl)formamido]-N-{[1-(phenoxymethyl)cyclopropyl]methyl}propanamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methoxyphenyl)piperazine
2-(2,5-dimethoxyphenyl)-4-(1H-imidazol-1-ylmethyl)-5-methyl-1,3-oxazole
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
2-[5-(5-ethylpyrimidin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(1S,5R)-3-(pyrazin-2-yl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-cyclopentyl-2-(methylamino)-N-(3-phenylprop-2-yn-1-yl)pyridine-3-carboxamide
1-[3-(morpholin-4-yl)benzoyl]-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
4-cycloheptyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(1H-imidazol-1-ylmethyl)-2-[3-(4-methylphenoxymethyl)piperidin-1-yl]pyridine
2-{4-[(2R)-2-amino-3-(4-chlorophenyl)propanoyl]piperazin-1-yl}-N-ethylacetamide