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7-(cyclopropylmethyl)-2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
6-cyclopentyl-N,1-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
5-[4-(1H-indol-3-yl)butan-2-yl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(5-butylthiophen-2-yl)methyl]-1,2-dimethylpiperazine
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(furan-3-carbonyl)-1,4-diazepane
1,3,7-trimethyl-2-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-[({1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-(2-methoxyethyl)-1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
6-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-chloro-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-(carbamoylmethyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine-3-carboxamide
5-chloro-N-methyl-N-(quinolin-5-ylmethyl)thiophene-2-carboxamide
2-(5-{imidazo[1,2-a]pyrimidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
methyl(quinolin-6-ylmethyl)[(2,3,4-trimethoxyphenyl)methyl]amine
2-{[1-tert-butyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydrophthalazin-1-one
4-[(5,6-dimethylpyrimidin-4-yl)amino]-1-(4-methoxyphenyl)pyrrolidin-2-one
8-(4-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
(3R,4S)-4-cyclopropyl-1-[2-(dimethylamino)benzoyl]pyrrolidin-3-amine
5-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2-ethylpyrimidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-2-carboxamide
2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]quinoline
6-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
4-[(3-fluorophenyl)methyl]-1-(2-oxo-2H-chromene-3-carbonyl)-1,4-diazepan-5-one
[5-(1H-pyrazol-3-yl)-1H-indol-2-yl]methanol
3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-N-(1,2,4-thiadiazol-5-yl)benzamide
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydroquinazoline-2,4-dione
1-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}thiophen-2-yl)ethan-1-one
N-[1-(pyridin-3-yl)propan-2-yl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-{5-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-methyl-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N6-[furan-2-yl(phenyl)methyl]-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxyacetamide
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-N-(2-fluorophenyl)piperidine-1-carboxamide
2-ethyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
3-(5-{2-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N-(diphenylmethyl)-2-[(3-hydroxy-2-methylphenyl)formamido]acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
1-{3-[4-({[(2,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
2-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-[(1-{6-[(oxolan-2-ylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-[5-(3-cyclopropyl-1H-pyrazol-5-yl)-3-(1H-indol-3-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,6,8-trimethylquinoline-4-carboxamide