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N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-3,5-dimethyl-1H-indole-2-carboxamide
N-(furan-3-ylmethyl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
N-[(2-methoxyphenyl)methyl]-2-phenyl-N-(prop-2-en-1-yl)propanamide
2-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-[(dimethylamino)methyl]pyrrolidin-3-ol
3-[(dimethylamino)methyl]-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}pyrrolidin-3-ol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}azepan-4-amine
2-(2-methoxyethoxy)-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
9-(2-hydroxybutanoyl)-2-(oxan-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
1-(3-{4-[(trimethyl-1H-pyrazol-4-yl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
N-[(3S,4R)-4-propyl-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methanesulfonamide
5-(2,4,6-trimethylphenyl)pyridin-3-amine
6-oxo-N-(thiophen-3-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-4-methyl-N-[(1-methylpiperidin-3-yl)methyl]benzene-1-sulfonamide
3-[4-(benzyloxy)piperidine-1-carbonyl]piperidine-1-carboxamide
(4S,4aS,8aS)-4-phenyl-1-(1-propyl-1H-pyrazole-5-carbonyl)-decahydroquinolin-4-ol
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]acetamide
(4aS,7aR)-1-(2-ethoxyacetyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)oxane-4-carboxamide
4-{5-[3-(1H-imidazol-1-yl)pyrrolidine-1-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
3-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}-4-fluorobenzene-1-sulfonamide
(1R,5S,6R,7S)-N-ethyl-3-methyl-4-oxo-N-[2-(phenylsulfanyl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3S,5R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-{1-[3-(1H-imidazol-5-yl)phenyl]-1H-imidazol-2-yl}benzoic acid
8-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidine
4-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-chloro-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-6-fluoro-N,3-dimethylbenzamide
N-cyclopropyl-1-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]piperazine-2-carboxamide
N2-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
4-methoxy-2,3,6-trimethyl-N-[(1-methylpiperidin-3-yl)methyl]benzene-1-sulfonamide
2-ethoxy-5-{2-[(oxan-3-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(pyridin-3-ylmethyl)benzamide
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-methyl-1,4-diazepan-5-one
(1S,2R)-2-({[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)amino)cyclohexan-1-ol
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-1-(thiomorpholin-4-yl)ethan-1-one
methyl 6-(2-cyclopentylacetyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)urea
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
6-methoxy-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-3-methyl-1-benzofuran-2-carboxamide
3-({2-[(2-chlorophenyl)formamido]ethyl}carbamoyl)benzoic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-aminopyridine-4-carboxamide
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-(propan-2-yl)pyridine-4-carboxamide