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3-(4-fluorophenyl)-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}propanoic acid
2-(5-chloro-2-methoxypyridin-4-yl)-4,5-difluorophenol
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2,3-dihydro-1H-inden-2-amine
3-[(2-methylphenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-[3-fluoro-4-(trifluoromethyl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-N,N-dimethylpyrazin-2-amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
N-cyclopentyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
4-[(3-fluorophenyl)methyl]-3-{2-[4-(2-methoxyethoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)pyrrolidine-3-carboxamide
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-(2-phenylethyl)piperidine
4-{[(1-benzylpiperidin-3-yl)carbamoyl]amino}-2-chlorobenzamide
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
3-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrazine-2-carbonitrile
N-{[1-(cyclopropylmethyl)piperidin-3-yl]methyl}cyclohexanecarboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methoxyhexanamide
N-[4-fluoro-3-(2-methylpropanamido)phenyl]-2-(2-methoxyethyl)piperidine-1-carboxamide
1-[2-({[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
4-{3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]propoxy}benzamide
6-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2,3-dihydropyridazin-3-one
2-{4-[4-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}-6-methylpyridine-3-carboxamide
2-amino-6-(2,5-dimethoxyphenyl)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
1-[(furan-2-ylmethyl)carbamoyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
2-[2,5-dioxo-4-(2-phenylethyl)-4-(piperidin-4-yl)imidazolidin-1-yl]-N-ethylacetamide
2-[(1S,5R)-6-(4-chloro-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
[1-(2,6-diaminopyrimidin-4-yl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
N-(2-oxopyrrolidin-3-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-(piperidin-4-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-methyl-3-oxo-N-[(1S)-1-phenylethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2-hydroxyethyl)-8-[(4-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-methoxybenzoyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
2-(morpholin-3-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
5-{pyrazolo[1,5-a]pyrimidin-3-yl}thiophene-2-carboxylic acid
methyl 2-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-methylpyridine-3-carboxamide
2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-4-amine
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methylphenoxy)acetamide
2-(methoxymethyl)-1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine
5-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-(2-methylphenyl)pyrimidine
5-methyl-6-(4-methylpiperazine-1-carbonyl)-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
5-butyl-1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
3-methyl-1-(2-methylphenyl)-4-(2-propylpyrimidin-5-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide