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3-(1H-1,2,3-benzotriazol-1-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
1-(3-methoxyphenyl)-4-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetyl}piperazin-2-one
1-(furan-2-carbonyl)-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepane
1-[5-(azepan-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]-4-methyl-1,4-diazepane
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-benzyl-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,3-benzoxazole
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-ethyl-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-4,4,4-trifluorobutanamide
2-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-4-methyl-N-(pentan-3-yl)pyrimidine-5-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-[4-(methylsulfanyl)phenyl]-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
N-cycloheptyl-3-ethyl-N-[(3-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
2-(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)pyridine
N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
N-(pyridin-3-ylmethyl)-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
2-{4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
7-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanecarboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[4-(pyridin-3-yloxy)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
3-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-(3,5-dimethoxyphenyl)propanamide
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-2-(morpholin-3-yl)acetamide
6-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,3,5,6-tetramethylbenzamide
2-(2,5-dimethoxyphenyl)-N-(propan-2-yl)pyridine-4-carboxamide
1-{3-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
2-{[4-(2-fluoro-4,5-dimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
(1S,3R)-3-amino-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]cyclopentane-1-carboxamide
5-{2-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
6-(2-aminoethyl)-N-cyclobutyl-2-methylpyrimidin-4-amine
1-{3-[3-({[(2,4-difluorophenyl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
N-[2-(2-chlorophenyl)ethyl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-methoxyacetamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(pyridin-3-ylmethyl)azepan-4-yl]acetamide
5-(5-cyclopropyl-1,2-oxazol-3-yl)-3-(4-ethoxyphenyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(2S,4S)-4-(4-{2-[(dimethylamino)methyl]phenoxymethyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxylic acid
3-cyclopropyl-5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-1,2,4-triazole
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
propan-2-yl N-[1-(cyclopropanesulfonyl)azepan-3-yl]carbamate
N-(adamantan-1-ylmethyl)-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-one
1-[3-methyl-1-(pyridin-3-yl)butyl]-3-(1-methyl-1H-1,2,4-triazol-3-yl)urea