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{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(2,4-dimethylphenyl)-4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazine
(3R,4R)-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-ol
3-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N,N-dimethylpropanamide
5-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,7-dimethylpyrazolo[1,5-a]pyrimidine
2-[1-(cyclohexylmethyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
(4aR,7aS)-4-(1H-1,3-benzodiazol-2-ylmethyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{[(8-methoxyquinolin-5-yl)methyl](methyl)amino}-N-(1,3-thiazol-2-yl)propanamide
(3aR,6aR)-2-acetyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-methyl-4-{3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propoxy}piperidine
2-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-{3-oxo-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-3-[2-(1H-pyrazol-1-yl)phenyl]urea
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
(8R,9aS)-2-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
4-[(4-methylphenyl)methyl]-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
(1S,5R)-3-[(5-ethylpyridin-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
5-chloro-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
5-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-2-(propan-2-yl)pyrimidine
1-cyclohexyl-N-[(5-methylpyrazin-2-yl)methyl]piperidine-4-carboxamide
2-fluoro-N-methyl-N-(quinolin-5-ylmethyl)-5-sulfamoylbenzamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-4-methylbenzoic acid
1-tert-butyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]cyclohexanamine
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(thiophen-2-ylmethyl)piperidin-4-ol
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-amine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-(thiolan-3-yl)piperidin-4-amine
5-amino-3-(5-chloro-2,4-dimethoxyphenyl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
(2-methoxy-5-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}phenyl)methanol
2-(5-acetylthiophen-3-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-[(1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperidin-4-yl)methyl]morpholine
3-(4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-(6-cyanopyridin-3-yl)-3-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]urea
(3S,4S)-1-[(4-carbamoylphenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
ethyl 1-{3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanoyl}piperidine-3-carboxylate
1-[1-(2-methoxyethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
13-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-ethyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2,5,7-trimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-yl)methyl]acetamide