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1-[(1-methyl-1H-imidazol-2-yl)methyl]-2,2-bis(prop-2-en-1-yl)piperidine
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(trifluoromethyl)benzamide
1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
6-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)pyridin-2-amine
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-[(2,6-dimethylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
2-ethyl-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
(2S,6S)-6-butyl-1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-oxazole-4-carboxamide
5-methyl-1-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-5-phenylpiperidin-2-one
4-(1,3-benzoxazol-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[4-(4-chlorophenyl)piperazine-1-carbonyl]-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
3-[2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
1-[3-(3-methoxyphenyl)phenyl]-3-[3-(3-oxopiperazin-1-yl)propyl]urea
N-methyl-2-{3-[3-(3-propanoylphenyl)phenyl]-1H-pyrazol-1-yl}acetamide
1-benzyl-5-(1H-imidazol-1-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
4-[2-hydroxy-4-(methylsulfanyl)butanoyl]-1-[(3-methylphenyl)methyl]piperazin-2-one
N-(2-methoxyethyl)-3-(1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)benzamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-(2,4-dimethylphenyl)-3-[2-(2-methylphenyl)pyrrolidin-1-yl]-3-oxopropanamide
2-(1H-1,3-benzodiazol-1-yl)-1-[2-(2-phenylethyl)morpholin-4-yl]ethan-1-one
14-(3,5-dimethoxyphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}){[1-(trifluoromethyl)cyclopropyl]methyl}amine
(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
N-(furan-2-ylmethyl)-4-[(3R)-3-hydroxypyrrolidin-1-yl]pyridine-2-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(4-chloro-2-methylphenoxy)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-(1H-indol-3-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)-4-methoxypiperidine
{3-benzyl-1-[2-(pyridin-3-yl)quinoline-4-carbonyl]piperidin-3-yl}methanol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(4-methoxyphenyl)-5-methyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
2-{[2-(dimethylamino)ethyl](methyl)amino}-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
6-(3,5-dichloro-4-methylbenzoyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
[(3R,4R)-1-[(4-ethoxyphenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
(1r,4r)-4-{[2-(2,3-dihydro-1H-inden-1-yl)acetamido]methyl}cyclohexane-1-carboxylic acid
methyl 2-({2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)acetate
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
(2R,3R)-3-amino-1'-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methoxy-5-({4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}methyl)benzoic acid
1-[3-(morpholin-4-yl)propyl]-6-oxo-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
2-(1H-pyrazol-3-yl)-4-(trifluoromethyl)pyrimidine
3-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-N-methylpyridin-2-amine
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one