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N,2,3-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-7-carboxamide
6-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-4-yl}pyrimidin-4-ol
1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(propylsulfanyl)ethan-1-one
N-[(4-hydroxyphenyl)methyl]-1-phenyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-phenylacetamide
N-(3,4-difluorophenyl)-1-(quinoxaline-5-carbonyl)piperidin-3-amine
1-[3-(piperidin-3-yl)benzoyl]azocane
2-(methoxymethyl)-1-[(2-phenyl-1H-imidazol-4-yl)methyl]piperidine
1-(4-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-methyl-4-(5-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}thiophen-2-yl)but-3-yn-2-ol
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-4-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylimidazo[1,2-a]pyridine-6-carboxamide
2-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-6-methoxyphenol
N-benzyl-5-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}pyrimidin-2-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2,5,7-trimethyl-N-(oxan-4-ylmethyl)quinoline-4-carboxamide
2-{9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)pyridin-2-amine
3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}azetidin-3-yl)pyridine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]amine
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-4-methyl-1H-imidazole
3-(2-methoxyethyl)-3-methyl-1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)urea
2-(2-aminoethyl)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methylquinazolin-4-amine
(2-{2-methoxy-6-[(4-methoxypiperidin-1-yl)methyl]phenoxy}ethyl)dimethylamine
2-(4-methyl-6-{[(2-propyl-1,3-thiazol-4-yl)methyl]amino}pyrimidin-2-yl)phenol
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2-methyl-1-benzofuran-5-carboxamide
[2-(azepan-1-yl)ethyl](ethyl)[(1-methyl-1H-imidazol-5-yl)methyl]amine
[(2,2-dimethyloxan-4-yl)methyl]({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl})amine
N-benzyl-N-ethyl-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-1,4-oxazepan-6-ol
2-(1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
ethyl 4-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}piperidine-1-carboxylate
5-ethyl-1'-[(3-methylquinoxalin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-pyrazol-1-yl)benzamide
6-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-(2-hydroxy-2-phenylethyl)-N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
7-(2,3-dimethoxyphenyl)-4-[(3-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(3S,4R)-1-[2-(2,3-difluorophenyl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1H-pyrrole-3-carboxamide
N-[(1-cyclopentanecarbonylpiperidin-3-yl)methyl]-4-methoxybenzene-1-sulfonamide
3-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
N4-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-methylpyrimidine-2,4-diamine
(2E)-3-(3-fluorophenyl)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)prop-2-enamide
N-[3-(1-tert-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]acetamide
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-ethoxypyridine
methyl 4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
(2S,4R)-4-{2-[benzyl(methyl)amino]acetamido}-1-(2-hydroxyethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide