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N-[2-(3,4-dimethoxyphenyl)ethyl]-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]amino}-1-(3-phenylpropyl)pyrrolidin-2-one
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-5-methyl-1,3,4-oxadiazol-2-amine
8-[(2-aminopyridin-3-yl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)ethan-1-ol
N-[(2S)-1-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-oxopropan-2-yl]acetamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-hydroxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(2H-1,3-benzodioxol-4-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
2,3-dimethyl-7-[3-(pyridin-2-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[4-(2-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethoxy)phenyl]propanamide
pyridin-2-yl(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanol
N-[2-(1H-indol-3-yl)ethyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
3-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-5-methoxy-3,4-dihydroquinazolin-4-one
(3R,4R)-4-ethyl-1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]piperidine-3,4-diol
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzamide
4-hydroxy-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-(4-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
2-(2-methylpropyl)-6-{thieno[2,3-d]pyrimidin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-[5-(1,3-dihydroxypropan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
methyl({2-[(2-methylpyridin-4-yl)oxy]hex-5-en-1-yl})(pyrazin-2-ylmethyl)amine
4-[5-(2,6-dimethoxypyridine-3-carbonyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-[(3S)-3-ethylmorpholin-4-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-benzyl-9-[2-oxo-2-(piperazin-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-[(3R,4S)-4-cyclopropyl-1-[(4-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl]-2-hydroxyacetamide
N-{[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
4-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-1-phenylpiperazin-2-one
2-(2-ethoxyethoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
8-chloro-2-(furan-2-yl)-4-[2-(methoxymethyl)piperidine-1-carbonyl]quinoline
(2S,3S)-2-{[1-(2-fluorophenyl)propan-2-yl]amino}-3-methylpentan-1-ol
2-{4-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenoxy}ethan-1-ol
methyl 4-{[3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}benzoate
3-{[(1-phenylpiperidin-4-yl)amino]methyl}piperidin-3-ol
2-[(3,3-dimethylcyclohexyl)amino]hexan-1-ol
2-{[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]methyl}-5-methoxy-4H-pyran-4-one
(3aS,7aR)-5-methyl-2-{[5-(4-methylphenyl)furan-2-yl]methyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-(5-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-2-methoxyphenyl)morpholine
(1S,5R)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S)-2-({2-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)-3-methylbutanoate
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-(1-methoxypropan-2-yl)-3-{[(4-methyl-1,3-thiazol-2-yl)methyl]sulfamoyl}benzamide
1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)spiro[azepane-4,2'-chromene]
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetamide
2-(4-hydroxyphenyl)-N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)acetamide
4-[(2-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine